SCHEMBL26439743

SCHEMBL26439743

Bc1ccc(C(F)(F)F)c2nccnc12

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NCF1 P14598 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
ALOX15 P16050 1/20 0.33
TSHR P16473 1/20 0.33
MAPK1 P28482 1/20 0.33
HIF1A Q16665 1/20 0.33
HSD17B10 Q99714 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
KIF11 P52732 2/20 0.32
PARP1 P09874 1/20 0.32
SLC40A1 Q9NP59 2/20 0.31
DYRK3 O43781 1/20 0.31
PRKD3 O94806 1/20 0.31
MAP4K4 O95819 1/20 0.31
CDK1 P06493 1/20 0.31
CDK2 P24941 1/20 0.31
FLT4 P35916 1/20 0.31
CSNK1D P48730 1/20 0.31
CLK2 P49760 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13626425 0.79 KDM4E (0.35) CYP3A4ALOX15TSHRHIF1ATDP1
SCHEMBL18892375 0.77 SLC40A1 (0.49) NCF1KIF11PARP1SLC40A1
SCHEMBL28083151 0.77 NCF1 (0.41) NCF1CYP1A2CYP3A4ALOX15TSHR
SCHEMBL19864754 0.77 PSMD14 (0.37) NCF1CYP1A2CYP3A4ALOX15TSHR
SCHEMBL18980694 0.75 NOTUM (0.35) NCF1CYP1A2CYP3A4ALOX15TSHR
SCHEMBL29722314 0.75 NOTUM (0.35) NCF1CYP1A2CYP3A4ALOX15TSHR
SCHEMBL21890801 0.68 IDO1 (0.43) SLC40A1DYRK3PRKD3MAP4K4CDK1
SCHEMBL13494774 0.67 CA2 (0.35) CYP1A2CYP3A4ALOX15TSHRHIF1A
SCHEMBL10840576 0.67 MAPT (0.48) NCF1CYP1A2CYP3A4ALOX15TSHR
SCHEMBL19864661 0.66 TLR7 (0.38) NCF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3844159-B1 NOVEL PYRROLIDINYL AMIDE COMPOUNDS FOR THE TREATMENT OF AUTOIMMUNE DISEASE HOFFMANN LA ROCHE (CH) 2023-05-03 EP disclosed