SCHEMBL2651898

SCHEMBL2651898

N#Cc1c(-c2ccccc2F)ccc(F)c1Br

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 4/20 0.41
ADORA2A P29274 3/20 0.41
ADORA2B P29275 2/20 0.38
ALDH1A1 P00352 6/20 0.38
KDM4E B2RXH2 4/20 0.38
HPGD P15428 4/20 0.38
GAA P10253 2/20 0.38
GLA P06280 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
CUL4A Q13619 1/20 0.37
GRIA2 P42262 1/20 0.35
GRIA4 P48058 1/20 0.35
HSD17B10 Q99714 3/20 0.35
MAPK1 P28482 2/20 0.35
CYP11B1 P15538 1/20 0.34
CYP11B2 P19099 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
RXFP1 Q9HBX9 1/20 0.34
PDE10A Q9Y233 1/20 0.33
MEN1 O00255 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6695094 0.81 ADORA1 (0.40) ADORA1ADORA2AADORA2BALDH1A1KDM4E
SCHEMBL2569036 0.79 ADORA1 (0.46) ADORA1ADORA2AADORA2BALDH1A1KDM4E
SCHEMBL16680707 0.76 TRPV4 (0.39) ALDH1A1KDM4EHPGDGAAHSD17B10
SCHEMBL2650101 0.74 ADORA1 (0.47) ADORA1ADORA2AADORA2BALDH1A1KDM4E
SCHEMBL2652911 0.73 ADORA1 (0.39) ADORA1ADORA2AADORA2BALDH1A1KDM4E
SCHEMBL28148660 0.73 ACHE (0.45) ADORA1ADORA2AADORA2BALDH1A1KDM4E
SCHEMBL2650208 0.72 GABRA5 (0.45) ADORA1ADORA2AADORA2BALDH1A1KDM4E
SCHEMBL2575063 0.72 ALDH1A1 (0.40) ADORA1ADORA2AADORA2BALDH1A1KDM4E
SCHEMBL19062287 0.72 ALDH1A1 (0.46) ADORA1ADORA2AADORA2BALDH1A1KDM4E
SCHEMBL16556066 0.69 TRPV4 (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004065388-A1 FLUOROIMIDAZOPYRIMIDINES AS GABA-A ALPHA 2/3 LIGANDS FOR DEPRESSION/ANXIETY MERCK SHARP & DOHME LIMITED (GB) 2004-08-05 WO disclosed