SCHEMBL2652111

SCHEMBL2652111

N#Cc1ccccc1C([O])OCc1ccccc1Br

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.41
TSHR P16473 1/20 0.36
ALDH1A1 P00352 2/20 0.35
MAOB P27338 1/20 0.35
PARP10 Q53GL7 1/20 0.35
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
SGMS2 Q8NHU3 1/20 0.34
FFAR1 O14842 2/20 0.33
MMP1 P03956 1/20 0.33
MMP2 P08253 1/20 0.33
MMP9 P14780 1/20 0.33
MMP12 P39900 1/20 0.33
FFAR4 Q5NUL3 1/20 0.33
CYP1A1 P04798 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP1B1 Q16678 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.32
KDM4E B2RXH2 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2652551 0.89 FFAR1 (0.41) TSHRALDH1A1MAOBNPC1RAB9A
SCHEMBL2651003 0.84 IDO1 (0.40) IDO1ALDH1A1MAOBPARP10NPC1
SCHEMBL2652007 0.84 TSHR (0.43) TSHRALDH1A1MAOBKDM4E
SCHEMBL2652010 0.84 IDO1 (0.40) IDO1MAOBNPC1RAB9A
SCHEMBL2650713 0.84 MAPK14 (0.37) TSHRALDH1A1NPC1RAB9ASGMS2
SCHEMBL2650913 0.82 IDO1 (0.50) IDO1TSHRALDH1A1PARP10NPC1
SCHEMBL2651078 0.81 IDO1 (0.44) IDO1ALDH1A1MAOBSMN1; SMN2
SCHEMBL2650110 0.81 TP53 (0.41) TSHRALDH1A1MAOBSGMS2FFAR1
SCHEMBL2650879 0.80 ALDH1A1 (0.48) TSHRALDH1A1MAOBSGMS2CYP1A2
SCHEMBL2650744 0.77 MAPK14 (0.37) TSHRALDH1A1SGMS2FFAR1MMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1404335-A1 AMINO NICOTINATE DERIVATIVES AS GLUCOKINASE (GLK) MODULATORS Astrazeneca AB (SE) 2004-04-07 EP disclosed
WO-2003000267-A1 AMINO NICOTINATE DERIVATIVES AS GLUCOKINASE (GLK) MODULATORS ASTRAZENECA AB (SE) 2003-01-03 WO disclosed