SCHEMBL26517604

SCHEMBL26517604

COc1cc(F)ccc1-c1nnc(N)c2ccncc12

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
UGCG Q16739 1/20 0.39
SCN9A Q15858 3/20 0.39
GPBAR1 Q8TDU6 8/20 0.39
PIP4K2A P48426 1/20 0.38
FYN P06241 2/20 0.38
CDK2 P24941 1/20 0.38
GSK3B P49841 1/20 0.38
KCNH2 Q12809 2/20 0.37
GRM5 P41594 1/20 0.37
PDE2A O00408 1/20 0.37
PDE4D Q08499 1/20 0.37
PDE3A Q14432 1/20 0.37
PDE10A Q9Y233 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24855740 0.82 EP300 (0.40) GPBAR1FYN
SCHEMBL31673746 0.81 MAOA (0.37) SCN9AFYN
SCHEMBL27355385 0.77 SCN9A (0.44) SCN9A
SCHEMBL24855382 0.76 EP300 (0.40) GPBAR1
SCHEMBL26516215 0.75 MGAT2 (0.41) CDK2GSK3B
SCHEMBL25857602 0.75 AMY1A (0.39) UGCGSCN9AFYN
SCHEMBL26517619 0.73 CLK1 (0.37) GSK3B
SCHEMBL31359797 0.72 CDK9 (0.38) CDK2GSK3BKCNH2
SCHEMBL24379596 0.72 SCN9A (0.40) SCN9A
SCHEMBL25857608 0.71 SCN9A (0.33) UGCGSCN9AFYNGRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023194964-A1 FUSED PYRIDAZINE DERIVATIVES AS NLRP3 INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2023-10-12 WO disclosed