SCHEMBL26547900

SCHEMBL26547900

CC(C)Nc1cc(-c2cccnc2)[nH]n1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 1/20 0.55
CYP3A4 P08684 3/20 0.50
ALDH1A1 P00352 2/20 0.50
CYP1A2 P05177 2/20 0.50
TNIK Q9UKE5 2/20 0.49
FLT3 P36888 1/20 0.47
HPGDS O60760 1/20 0.47
CYP2A6 P11509 4/20 0.45
CYP2E1 P05181 2/20 0.45
CYP2B6 P20813 2/20 0.45
ALK Q9UM73 1/20 0.44
DYRK1A Q13627 6/20 0.42
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
CLK2 P49760 5/20 0.41
CLK3 P49761 5/20 0.41
MAP2K4 P45985 1/20 0.40
PRKAB2 O43741 1/20 0.40
PRKAG1 P54619 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25431149 0.83 RAB9A (0.53) CHEK1ALDH1A1TNIK
SCHEMBL26547901 0.81 ROCK2 (0.46) ALDH1A1TNIKPRKAB2PRKAG1PRKAA2
SCHEMBL30579362 0.77 CYP3A4 (0.54) CHEK1CYP3A4ALDH1A1CYP1A2TNIK
SCHEMBL10022326 0.77 CYP3A4 (0.54) CHEK1CYP3A4ALDH1A1CYP1A2TNIK
SCHEMBL2318425 0.74 CYP3A4 (0.59) CHEK1CYP3A4ALDH1A1CYP1A2TNIK
SCHEMBL26551519 0.73 FLT3 (0.62) CYP3A4ALDH1A1CYP1A2FLT3CYP2A6
SCHEMBL3078162 0.73 CYP3A4 (0.89) CYP3A4ALDH1A1CYP1A2HPGDSCYP2A6
SCHEMBL28207587 0.73 ALDH1A1 (0.61) CHEK1CYP3A4ALDH1A1CYP1A2HPGDS
SCHEMBL9564384 0.72 FLT3 (0.48) CYP3A4ALDH1A1CYP1A2FLT3CYP2A6
SCHEMBL30872899 0.72 CYP3A4 (0.51) CHEK1CYP3A4ALDH1A1CYP1A2TNIK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023196975-A1 COMPOUNDS THAT INTERACT WITH RAS SUPERFAMILY PROTEINS FOR TREATMENT OF CANCERS, INFLAMMATORY DISEASES, RASOPATHIES, AND FIBROTIC DISEASE SHY THERAPEUTICS, LLC (US) 2023-10-12 WO disclosed