SCHEMBL265605

SCHEMBL265605

N[C@@H](CC1CCCCC1)C(=O)NCC(=O)NCC(=O)N(C(=O)c1ccco1)[C@@H](CCCN1CCCCC1)C(=O)NCc1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 1/20 0.39
OPRM1 P35372 4/20 0.35
MMP1 P03956 3/20 0.35
MMP2 P08253 1/20 0.35
MMP3 P08254 1/20 0.35
CYP2D6 P10635 2/20 0.35
TP53 P04637 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
TSHR P16473 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
FCER2 P06734 2/20 0.35
BMP1 P13497 1/20 0.35
OPRK1 P41145 3/20 0.34
REN P00797 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
OPRD1 P41143 2/20 0.34
HSD17B10 Q99714 1/20 0.34
MEN1 O00255 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL265370 0.93 MMP1 (0.39) CCR5MMP1MMP2MMP3CYP2D6
Hydrochloric Acid SCHEMBL266228 0.92 MMP1 (0.38) CCR5MMP1MMP2MMP3CYP2D6
SCHEMBL1450242 0.88 MMP1 (0.39) CCR5OPRM1MMP1MMP2MMP3
SCHEMBL1449025 0.86 REN (0.42) CCR5MMP1MMP2MMP3REN
SCHEMBL5574185 0.81 HPGD (0.40) CCR5OPRM1MMP1MMP2FCER2
SCHEMBL1449086 0.77 SLC6A2 (0.41) MMP1MMP2MMP3OPRK1REN
SCHEMBL313931 0.77 CTSS (0.48) MMP1MMP2MMP3FCER2REN
SCHEMBL272047 0.77 CTSS (0.48) MMP1MMP2MMP3FCER2REN
SCHEMBL1449333 0.76 MMP1 (0.39) MMP1MMP2MMP3TDP1REN
SCHEMBL1449031 0.76 MMP3 (0.35) MMP1MMP2MMP3CYP2D6TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8133864-B2 PAR-2 agonist KOWA COMPANY, LTD. (JP) 2012-03-13 US claimed
EP-1864994-B1 PAR-2 AGONIST KOWA CO (JP) 2011-10-26 EP claimed
US-8133864-B2 PAR-2 agonist KOWA COMPANY, LTD. (JP) 2012-03-13 US disclosed