SCHEMBL2657582

SCHEMBL2657582

C[C@@H](N)c1ccc2c(c1)ncn2-c1ccc(F)c(-c2cccnc2F)c1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.39
GABRA1 P14867 3/20 0.37
HPGD P15428 2/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2C9 P11712 1/20 0.37
MAPK1 P28482 1/20 0.37
CYP2C19 P33261 1/20 0.37
FGFR1 P11362 7/20 0.37
CTSD P07339 5/20 0.36
BACE1 P56817 5/20 0.36
BACE2 Q9Y5Z0 5/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
ALDH1A1 P00352 1/20 0.34
MAPT P10636 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
REN P00797 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2657860 0.90 GABRA1 (0.46) THRBGABRA1HPGDCYP1A2CYP2C9
SCHEMBL2658067 0.88 GABRA1 (0.48) THRBGABRA1HPGDCYP1A2CYP2C9
SCHEMBL2659305 0.88 GABRA1 (0.48) THRBGABRA1HPGDCYP1A2CYP2C9
SCHEMBL2659103 0.85 FGFR1 (0.43) THRBGABRA1HPGDCYP1A2CYP2C9
SCHEMBL3767124 0.85 GABRA1 (0.43) GABRA1HPGDFGFR1CTSDBACE1
SCHEMBL2651205 0.85 GABRA1 (0.43) GABRA1HPGDFGFR1CTSDBACE1
SCHEMBL2654319 0.85 GABRA1 (0.43) GABRA1HPGDFGFR1CTSDBACE1
SCHEMBL2656812 0.83 FGFR1 (0.39) THRBGABRA1HPGDCYP1A2CYP2C9
SCHEMBL2339374 0.79 GABRA1 (0.60) THRBGABRA1HPGDCYP1A2CYP2C9
SCHEMBL2669578 0.79 THRB (0.44) THRBGABRA1HPGDCYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010055125-A1 BENZIMIDAZOLE DERIVATIVES AND THEIR USE FOR MODULATING THE GABAA RECEPTOR COMPLEX NEUROSEARCH A/S (DK) 2010-05-20 WO claimed
WO-2010055125-A1 BENZIMIDAZOLE DERIVATIVES AND THEIR USE FOR MODULATING THE GABAA RECEPTOR COMPLEX NEUROSEARCH A/S (DK) 2010-05-20 WO disclosed