SCHEMBL2659103

SCHEMBL2659103

C[C@@H](N)c1ccc2c(c1)ncn2-c1ccc(F)c(-c2ccccc2Cl)c1

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
FGFR1 P11362 8/20 0.43
THRB P10828 1/20 0.39
NR1I2 O75469 1/20 0.37
TP53 P04637 1/20 0.37
HPGD P15428 6/20 0.37
ALDH1A1 P00352 1/20 0.35
GABRA1 P14867 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2C9 P11712 1/20 0.35
MAPK1 P28482 1/20 0.35
CYP2C19 P33261 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2657860 0.88 GABRA1 (0.46) FGFR1THRBHPGDALDH1A1GABRA1
SCHEMBL2657582 0.85 THRB (0.39) FGFR1THRBHPGDALDH1A1GABRA1
SCHEMBL2656812 0.83 FGFR1 (0.39) FGFR1THRBHPGDALDH1A1GABRA1
SCHEMBL2657177 0.82 GABRA1 (0.51) FGFR1NR1I2TP53HPGDGABRA1
SCHEMBL2658067 0.82 GABRA1 (0.48) FGFR1THRBHPGDALDH1A1GABRA1
SCHEMBL2659305 0.82 GABRA1 (0.48) FGFR1THRBHPGDALDH1A1GABRA1
SCHEMBL1616703 0.81 GABRA1 (0.46) FGFR1HPGDGABRA1
SCHEMBL2657910 0.79 GABRA1 (0.57) FGFR1THRBNR1I2TP53HPGD
SCHEMBL2669578 0.79 THRB (0.44) FGFR1THRBHPGDALDH1A1GABRA1
SCHEMBL2658314 0.79 SIK1 (0.40) FGFR1THRBTP53HPGDALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010055125-A1 BENZIMIDAZOLE DERIVATIVES AND THEIR USE FOR MODULATING THE GABAA RECEPTOR COMPLEX NEUROSEARCH A/S (DK) 2010-05-20 WO claimed