SCHEMBL2669320

SCHEMBL2669320

CCOC(=O)C(N)CC1CCC(F)(F)CC1

nearest known ligand 0.35

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
METAP2 P50579 2/20 0.35
NAAA Q02083 1/20 0.34
ASAH1 Q13510 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.33
CYP2D6 P10635 1/20 0.31
GAA P10253 1/20 0.31
TRPM8 Q7Z2W7 1/20 0.31
ALOX15 P16050 1/20 0.31
REN P00797 1/20 0.30
TSHR P16473 1/20 0.30
JAK2 O60674 1/20 0.30
JAK1 P23458 1/20 0.30
TYK2 P29597 1/20 0.30
JAK3 P52333 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12023171 0.86 NAAA (0.37) NAAAASAH1REN
SCHEMBL28270788 0.85 L3MBTL1 (0.39) METAP2L3MBTL1CYP2D6GAAALOX15
SCHEMBL12201811 0.84 CYP3A4 (0.35) METAP2NAAAASAH1L3MBTL1CYP2D6
SCHEMBL1066592 0.82 METAP2 (0.42) METAP2L3MBTL1CYP2D6GAAALOX15
SCHEMBL28785091 0.82 METAP2 (0.42) METAP2L3MBTL1CYP2D6GAAALOX15
SCHEMBL20543740 0.82 METAP2 (0.45) METAP2CYP2D6RENTSHR
SCHEMBL24548571 0.80 EPHX2 (0.34) NAAAASAH1
SCHEMBL21118051 0.80 METAP2 (0.47) METAP2RENTSHR
SCHEMBL9555738 0.80 METAP2 (0.47) METAP2RENTSHR
SCHEMBL13836892 0.80 METAP2 (0.47) METAP2RENTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240277795-A1 INHIBITORS OF CYSTEINE PROTEASES AND METHODS OF USE THEREOF PARDES BIOSCIENCES INC (US) 2024-08-22 US disclosed
EP-4387980-A1 INHIBITORS OF CYSTEINE PROTEASES AND METHODS OF USE THEREOF Pardes Biosciences, Inc. (US) 2024-06-26 EP disclosed
WO-2023023631-A1 INHIBITORS OF CYSTEINE PROTEASES AND METHODS OF USE THEREOF Pardes Biosciences, Inc. (US) 2023-02-23 WO disclosed
WO-2023023631-A1 INHIBITORS OF CYSTEINE PROTEASES AND METHODS OF USE THEREOF Pardes Biosciences, Inc. (US) 2023-02-23 WO disclosed
US-8034822-B2 Glucokinase activators TAKEDA SAN DIEGO, INC. (US) 2011-10-11 US disclosed
US-8034822-B2 Glucokinase activators TAKEDA SAN DIEGO, INC. (US) 2011-10-11 US disclosed
WO-2007104034-A2 GLUCOKINASE ACTIVATORS TAKEDA SAN DIEGO, INC. (US) 2007-09-13 WO disclosed
US-20070213349-A1 GLUCOKINASE ACTIVATORS TAKEDA SAN DIEGO, INC. 2007-09-13 US disclosed
US-20070213349-A1 GLUCOKINASE ACTIVATORS TAKEDA SAN DIEGO, INC. 2007-09-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240277795-A1 INHIBITORS OF CYSTEINE PROTEASES AND METHODS OF USE THEREOF CTRL, CPN1, CTSL METAP2 225/4885NAAA 551/4885ASAH1 1824/4885
US-20070213349-A1 GLUCOKINASE ACTIVATORS GCK, GCKR, GALK1 METAP2 1519/4885NAAA 996/4885ASAH1 780/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.