SCHEMBL26783003

SCHEMBL26783003

CC(C#N)C12CC(C1)C(NC(=O)OC(C)(C)C)C2

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CTSK P43235 10/20 0.39
CTSL P07711 3/20 0.38
CTSS P25774 7/20 0.37
CTSB P07858 2/20 0.36
HSD11B1 P28845 1/20 0.35
NFKB1 P19838 1/20 0.34
NFKB2 Q00653 1/20 0.34
RELA Q04206 1/20 0.34
KDM1A O60341 1/20 0.34
BTK Q06187 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26782822 0.74 CTSK (0.40) CTSKCTSLCTSSCTSBHSD11B1
SCHEMBL23281289 0.72 NFKB1 (0.40) CTSKHSD11B1NFKB1NFKB2RELA
SCHEMBL26783023 0.72 CTSL (0.39) CTSKCTSLCTSSCTSBNFKB1
SCHEMBL24337068 0.71 BTK (0.39) CTSKHSD11B1NFKB1NFKB2RELA
SCHEMBL21503946 0.71 CTSL (0.40) CTSKCTSLCTSSCTSB
SCHEMBL23900563 0.71 BTK (0.44) CTSKHSD11B1NFKB1NFKB2RELA
SCHEMBL23625485 0.71 BTK (0.44) CTSKHSD11B1NFKB1NFKB2RELA
SCHEMBL23562417 0.71 HSD11B1 (0.47) CTSKHSD11B1NFKB1NFKB2RELA
SCHEMBL24543130 0.71 BTK (0.44) CTSKHSD11B1NFKB1NFKB2RELA
SCHEMBL23562416 0.70 HSD11B1 (0.49) CTSKHSD11B1NFKB1NFKB2RELA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3810116-B1 NOVEL SUBSTITUTED [1.1.1] BICYCLO COMPOUNDS AS INDOLEAMINE 2,3-DIOXYGENASE INHIBITORS MERCK SHARP & DOHME LLC (US) 2023-11-15 EP disclosed