SCHEMBL26909780

SCHEMBL26909780

NC(=O)C(Cc1ccc(-c2ccccc2)cc1)NC(=O)O

nearest known ligand 0.58

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HPGDS O60760 5/20 0.58
MME P08473 11/20 0.55
ACE2 Q9BYF1 9/20 0.55
ACE P12821 8/20 0.52
CPA1 P15085 7/20 0.52
SRR Q9GZT4 2/20 0.51
PSAT1 Q9Y617 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4348297 1.00 HPGDS (0.58) HPGDSMMEACE2ACECPA1
SCHEMBL9109075 0.91 HPGDS (0.56) HPGDSMME
SCHEMBL299180 0.85 CTSC (0.49) HPGDSMMEACE2ACECPA1
SCHEMBL28097066 0.85 HPGDS (0.47) HPGDSACE
SCHEMBL24899372 0.84 HPGDS (0.56) HPGDSMMEACE2ACECPA1
SCHEMBL2074867 0.84 CA1 (0.51) HPGDS
SCHEMBL16823433 0.84 HPGDS (0.53) HPGDSMMEACE2ACECPA1
SCHEMBL30995919 0.84 MME (0.55) HPGDSMMEACE2ACECPA1
SCHEMBL18262572 0.83 CA2 (0.49) HPGDSMME
SCHEMBL20397627 0.83 FPR2 (0.48) HPGDS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230391766-A1 1-(2-(4-CYCLOPROPYL-1H-1,2,3-TRIAZOL-1-YL)ACETYL)-4-HYDROXY-N-(BENZYL)PYRROLIDIN E-2-CARBOXAMIDE DERIVATIVES AS VHL INHIBITORS FOR THE TREATMENT OF ANEMIA AND CANCER GENENTECH, INC. (US) 2023-12-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230391766-A1 1-(2-(4-CYCLOPROPYL-1H-1,2,3-TRIAZOL-1-YL)ACETYL)-4-HYDROXY-N-(BENZYL)PYRROLIDIN E-2-CARBOXAMIDE DERIVATIVES AS VHL INHIBITORS FOR THE TREATMENT OF ANEMIA AND CANCER VHL, HIF1AN, EGLN2 HPGDS 98/4885MME 4519/4885ACE2 3593/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.