SCHEMBL2714933

SCHEMBL2714933

Cc1ccc(-c2ccc(CC(N)=O)nc2)cn1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 3/20 0.42
HTT P42858 1/20 0.40
CYP11B2 P19099 1/20 0.39
KCNH2 Q12809 1/20 0.39
ATM Q13315 1/20 0.39
ATR Q13535 1/20 0.39
ADRA2A P08913 2/20 0.39
ADRA2B P18089 2/20 0.39
ADRA2C P18825 2/20 0.39
IDO1 P14902 1/20 0.39
LGMN Q99538 1/20 0.38
PTGS2 P35354 1/20 0.38
BRD4 O60885 1/20 0.38
PRMT5 O14744 1/20 0.38
WDR77 Q9BQA1 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
PIK3CD O00329 1/20 0.37
PIK3CA P42336 1/20 0.37
PIK3CB P42338 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30440577 0.81 SRC (0.51) HTTKCNJ6KCNJ3MKNK1MKNK2
SCHEMBL19376938 0.81 MKNK1 (0.55) CYP11B2ALDH1A1MKNK1MKNK2
SCHEMBL19376930 0.80 CHEK2 (0.44) HDAC1HDAC6MKNK1MKNK2
SCHEMBL17675624 0.80 EGLN1 (0.41) CYP11B2KCNH2ATMPRMT5HDAC1
SCHEMBL1428296 0.79 ADRA2A (0.47) HTTADRA2AADRA2BADRA2CHDAC6
SCHEMBL28508293 0.77 MET (0.50) CYP11B2KCNH2ATMATRMKNK1
SCHEMBL30595305 0.77 HTT (0.46) HTTADRA2AADRA2BADRA2CALDH1A1
SCHEMBL15006455 0.77 HTT (0.46) HTTADRA2AADRA2BADRA2CALDH1A1
SCHEMBL25263472 0.77 PRMT5 (0.46) ADRA2AADRA2BADRA2CPTGS2PRMT5
SCHEMBL17675606 0.77 ADRB2 (0.41) KCNH2HDAC1HDAC6RAB9AMKNK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2445909-A1 DERIVATIVES OF 6,7-DIHYDRO-5H-IMIDAZO[1,2-a]IMIDAZOLE-3-CARBOXYLIC ACID AMIDES Boehringer Ingelheim International GmbH (DE) 2012-05-02 EP disclosed
WO-2010141273-A1 DERIVATIVES OF 6,7-DIHYDRO-5H-IMIDAZO[1,2-a]IMIDAZOLE-3-CARBOXYLIC ACID AMIDES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-12-09 WO disclosed