SCHEMBL2718367

SCHEMBL2718367

COCCc1c([N+](=O)[O-])ccc(N)c1N

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.44
ALDH1A1 P00352 5/20 0.44
LMNA P02545 2/20 0.41
TSHR P16473 2/20 0.40
TDP1 Q9NUW8 5/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
POLB P06746 2/20 0.39
CYP3A4 P08684 1/20 0.39
ALOX15 P16050 1/20 0.39
HTT P42858 1/20 0.38
MAPK1 P28482 2/20 0.38
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
PKM P14618 2/20 0.35
KDM4E B2RXH2 1/20 0.35
G6PD P11413 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6232035 0.91 ALDH1A1 (0.43) MAPTALDH1A1LMNATSHRTDP1
SCHEMBL14892862 0.88 MAPT (0.44) MAPTALDH1A1LMNATSHRTDP1
SCHEMBL14893069 0.80 ALDH1A1 (0.41) MAPTALDH1A1LMNATSHRTDP1
SCHEMBL6983628 0.80 ALDH1A1 (0.43) MAPTALDH1A1LMNATSHRTDP1
SCHEMBL17242666 0.79 TSHR (0.45) MAPTALDH1A1LMNATSHRTDP1
SCHEMBL25221130 0.79 MAPT (0.36) MAPTALDH1A1LMNATSHRTDP1
SCHEMBL9820274 0.79 ALDH1A1 (0.42) MAPTALDH1A1LMNATDP1MEN1
SCHEMBL17186886 0.79 ALDH1A1 (0.42) MAPTALDH1A1LMNATSHRTDP1
SCHEMBL5484250 0.79 TSHR (0.44) MAPTALDH1A1LMNATSHRTDP1
SCHEMBL2337048 0.78 POLB (0.47) MAPTALDH1A1LMNATSHRTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012059932-A1 2, 4 -DIAMINOPYRIMIDINE DERIVATIVES AS PROTEIN KINASE INHIBITORS AURIGENE DISCOVERY TECHNOLOGIES LIMITED (IN) 2012-05-10 WO disclosed