SCHEMBL2720271

SCHEMBL2720271

NC(=O)OC1(c2ccc(C(=O)CBr)cc2)CCC1

nearest known ligand 0.42

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 11/20 0.42
PTPN1 P18031 6/20 0.42
DRD2 P14416 6/20 0.34
DRD4 P21917 6/20 0.34
DRD3 P35462 6/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3803479 0.81 L3MBTL1 (0.47) DRD3
SCHEMBL15258665 0.81 MAPT (0.44)
SCHEMBL3813595 0.80 ALDH1A1 (0.36)
SCHEMBL17698403 0.78 ALDH1A1 (0.41)
SCHEMBL3812202 0.76 HSD11B1 (0.43) DRD2DRD4DRD3
SCHEMBL26135641 0.76 AKR1C1 (0.44) DRD3
SCHEMBL15258670 0.74 MAPT (0.46)
SCHEMBL4849593 0.73 PARP15 (0.41) GSK3B
SCHEMBL11289324 0.73 AKR1C1 (0.48)
SCHEMBL2720401 0.73 CA1 (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012061342-A2 SUBSTITUTED BENZO-IMIDAZO-PYRIDO-DIAZEPINE COMPOUNDS ARQULE, INC. (US) 2012-05-10 WO disclosed