SCHEMBL4849593

SCHEMBL4849593

N#Cc1ccc(C2(OC(N)=O)CCC2)cc1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PARP15 Q460N3 1/20 0.41
PARP10 Q53GL7 1/20 0.41
PARP2 Q9UGN5 1/20 0.41
CA1 P00915 2/20 0.40
CA2 P00918 2/20 0.40
CYP19A1 P11511 2/20 0.36
POLB P06746 1/20 0.36
LMNA P02545 1/20 0.36
IDO1 P14902 2/20 0.35
EPHX1 P07099 1/20 0.35
PGR P06401 1/20 0.34
NOS3 P29474 1/20 0.34
NOS1 P29475 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
MMP2 P08253 1/20 0.34
CTSC P53634 1/20 0.34
KCNH2 Q12809 1/20 0.34
GSK3B P49841 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17698403 0.80 ALDH1A1 (0.41) PARP10CYP19A1POLBLMNARAB9A
SCHEMBL3813595 0.79 ALDH1A1 (0.36) CA1CA2POLBLMNANPC1
SCHEMBL3812202 0.79 HSD11B1 (0.43)
SCHEMBL24616687 0.79 CA1 (0.35) CA1CA2CYP19A1LMNAPGR
SCHEMBL27920662 0.79 PGR (0.39) CA1CA2CYP19A1PGRNPC1
SCHEMBL26135641 0.78 AKR1C1 (0.44)
SCHEMBL1904598 0.78 CYP3A4 (0.34)
SCHEMBL16495248 0.77 PTGDR2 (0.41) CA1CA2CYP19A1LMNAMMP2
SCHEMBL1900928 0.76 RAB9A (0.36) LMNARAB9A
SCHEMBL24397821 0.76 SIGMAR1 (0.35) CA1CA2POLBLMNAPGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008070041-A2 INHIBITORS OF AKT ACTIVITY MERCK & CO., INC. (US) 2008-06-12 WO disclosed