SCHEMBL27299154

SCHEMBL27299154

COC(=O)C(N)c1ccc(N(C)C(C)C)nc1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 1/20 0.39
KLKB1 P03952 1/20 0.37
KLK1 P06870 1/20 0.37
TRPV1 Q8NER1 1/20 0.36
GAA P10253 1/20 0.33
KMT2A Q03164 1/20 0.32
MT-CO2 P00403 1/20 0.32
HCAR3 P49019 1/20 0.31
REN P00797 1/20 0.31
ROCK2 O75116 1/20 0.31
MCHR1 Q99705 1/20 0.31
GRM1 Q13255 1/20 0.31
AOC3 Q16853 1/20 0.30
ALDH1A1 P00352 1/20 0.30
VNN1 O95497 1/20 0.30
ESR1 P03372 1/20 0.30
ESR2 Q92731 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31473371 1.00 PDE10A (0.39) PDE10AKLKB1KLK1TRPV1GAA
SCHEMBL7252180 0.73 KMT2A (0.48) KMT2AMT-CO2ALDH1A1ESR1ESR2
SCHEMBL31473467 0.71 HCAR3 (0.41) PDE10AKLKB1KLK1TRPV1KMT2A
SCHEMBL27299149 0.71 HCAR3 (0.41) PDE10AKLKB1KLK1TRPV1KMT2A
SCHEMBL27299043 0.71 PDE4A (0.35) PDE10AAOC3
SCHEMBL22387918 0.71 PDE10A (0.37) PDE10A
SCHEMBL14658669 0.70 TRPV1 (0.55) TRPV1MT-CO2HCAR3AOC3
SCHEMBL14032514 0.70 L3MBTL1 (0.46) KMT2AMT-CO2ALDH1A1
SCHEMBL14660039 0.69 DGAT1 (0.47) TRPV1HCAR3
SCHEMBL31473426 0.69 HCAR3 (0.47) PDE10AKLKB1KLK1HCAR3GRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024029489-A1 KIT INHIBITORS, COMPOUNDS, PHARMACEUTICAL COMPOSITIONS, AND METHODS OF USE THEREOF MODULUS DISCOVERY, INC. (JP) 2024-02-08 WO disclosed