SCHEMBL2732401

SCHEMBL2732401

O=C(O)N1CCCC(c2nc(N=C(c3ccccc3)c3ccccc3)cc3[nH]cnc23)C1

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.37
HPGD P15428 1/20 0.37
MAP3K12 Q12852 6/20 0.37
PDE2A O00408 2/20 0.36
HSD11B1 P28845 2/20 0.36
PROKR1 Q8TCW9 3/20 0.35
NPC1 O15118 1/20 0.35
TP53 P04637 1/20 0.35
MAPT P10636 1/20 0.35
TSHR P16473 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
PDE3A Q14432 1/20 0.34
JAK2 O60674 1/20 0.34
JAK1 P23458 1/20 0.34
TYK2 P29597 1/20 0.34
JAK3 P52333 1/20 0.34
ADORA2A P29274 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2767593 0.66 CTNNB1 (0.35) ALDH1A1HPGDNPC1TP53MAPT
SCHEMBL27201572 0.65 HSD11B1 (0.64) ALDH1A1HSD11B1
SCHEMBL174319 0.64 L3MBTL1 (0.36) ALDH1A1HPGDPROKR1NPC1RAB9A
SCHEMBL2789326 0.62 AKR1C3 (0.49) HPGDMAPTSMN1; SMN2
SCHEMBL3312540 0.62 ALDH1A1 (0.62) ALDH1A1HPGDHSD11B1PROKR1NPC1
SCHEMBL28080532 0.62 JAK3 (0.52) JAK2JAK1TYK2JAK3
SCHEMBL23580775 0.62 BTK (0.35) ALDH1A1HPGD
SCHEMBL23580773 0.62 BTK (0.35) ALDH1A1HPGD
SCHEMBL2514536 0.62 HTR2B (0.61) SMN1; SMN2
SCHEMBL2520100 0.62 HTR2B (0.61) SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2632898-A1 HETEROCYCLIC TYROSINE KINASE INHIBITORS Biogen Idec MA Inc. (US) 2013-09-04 EP disclosed
WO-2012058645-A1 HETEROCYCLIC TYROSINE KINASE INHIBITORS BIOGEN IDEC MA INC. (US) 2012-05-03 WO disclosed