SCHEMBL27324835

SCHEMBL27324835

c1ccc(-c2noc(CN3CCNCC3)n2)cc1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.72
CYP2D6 P10635 2/20 0.72
NPC1 O15118 3/20 0.66
RAB9A P51151 3/20 0.66
LMNA P02545 6/20 0.64
HTT P42858 2/20 0.64
NPSR1 Q6W5P4 1/20 0.64
MAPK1 P28482 2/20 0.63
ALDH1A1 P00352 4/20 0.62
KMT2A Q03164 3/20 0.62
MEN1 O00255 2/20 0.62
L3MBTL1 Q9Y468 2/20 0.62
CASP1 P29466 1/20 0.62
CASP7 P55210 1/20 0.62
MAPT P10636 3/20 0.61
SMN1; SMN2 Q16637 3/20 0.61
TSHR P16473 1/20 0.61
HSD17B10 Q99714 1/20 0.61
POLB P06746 2/20 0.57
PKM P14618 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24326609 0.86 RAB9A (0.76) KCNH2CYP2D6NPC1RAB9ALMNA
SCHEMBL23958379 0.81 CYP2D6 (0.92) KCNH2CYP2D6NPC1RAB9ALMNA
SCHEMBL31532358 0.80 KCNH2 (0.60) KCNH2CYP2D6NPC1RAB9ALMNA
SCHEMBL26887340 0.78 SPHK2 (0.58) KCNH2CYP2D6NPC1RAB9ALMNA
Hydrochloric Acid SCHEMBL15231570 0.77 S1PR1 (0.45) KCNH2CYP2D6NPC1RAB9ALMNA
SCHEMBL44702 0.76 KCNH2 (0.44) KCNH2CYP2D6NPC1RAB9ALMNA
SCHEMBL17115053 0.75 FAAH (0.48) KCNH2CYP2D6HTTALDH1A1KMT2A
SCHEMBL14703941 0.74 RAB9A (0.74) KCNH2CYP2D6NPC1RAB9ALMNA
SCHEMBL14890146 0.74 MAPT (0.78) KCNH2CYP2D6NPC1RAB9ALMNA
SCHEMBL2089284 0.73 NOTUM (0.68) KCNH2CYP2D6NPC1RAB9AMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024088922-A1 HETEROCYCLIC COMPOUNDS AS INHIBITORS OF MONOACYLGLYCEROL LIPASE (MAGL) F. HOFFMANN-LA ROCHE AG (CH) 2024-05-02 WO disclosed