SCHEMBL27344682

SCHEMBL27344682

CC(C)(C)Oc1ccccc1-c1ccccc1.[SiH3]Cl

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 1/20 0.43
ADRB2 P07550 6/20 0.42
ADRB1 P08588 2/20 0.42
MAPK1 P28482 2/20 0.42
TP53 P04637 1/20 0.42
RAB9A P51151 1/20 0.42
NCOA1 Q15788 1/20 0.42
NCOA3 Q9Y6Q9 1/20 0.42
TDP1 Q9NUW8 2/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
LMNA P02545 1/20 0.41
CYP2A6 P11509 1/20 0.40
HRH1 P35367 1/20 0.40
ALDH1A1 P00352 2/20 0.38
KDM4E B2RXH2 3/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
PTGS2 P35354 1/20 0.37
ADRA2A P08913 1/20 0.36
ADRA2B P18089 1/20 0.36
ADRA2C P18825 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8017279 0.96 HTR7 (0.46) HTR7ADRB2ADRB1MAPK1TP53
SCHEMBL27515199 0.94 HTR7 (0.44) HTR7ADRB2ADRB1MAPK1TP53
Hydrogen Sulfide SCHEMBL27894468 0.90 HTR7 (0.42) HTR7ADRB2ADRB1MAPK1TP53
SCHEMBL12355661 0.83 CA12 (0.39) HTR7MAPK1L3MBTL1ALDH1A1KDM4E
SCHEMBL22174608 0.80 HTR7 (0.43) HTR7ADRB2ADRB1MAPK1TP53
SCHEMBL27460371 0.77 ADRB2 (0.46) HTR7ADRB2ADRB1MAPK1TP53
SCHEMBL27335556 0.77 L3MBTL1 (0.49) ADRB2ADRB1MAPK1NCOA1NCOA3
SCHEMBL28340902 0.77 LMNA (0.46) ADRB2ADRB1MAPK1TDP1L3MBTL1
SCHEMBL7049020 0.77 TAAR1 (0.46) ADRB2MAPK1TP53RAB9A
SCHEMBL12164572 0.76 KIF11 (0.42) MAPK1NCOA1NCOA3L3MBTL1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1052229-C 7-deoxy-taxol and pharmaceutical composition thereof BRISTOL MYERS SQUIBB CO (US) 2000-05-10 CN disclosed
CN-1051309-C Fluoro taxol BRISTOL MYERS SQUIBB CO (US) 2000-04-12 CN disclosed
CN-1085553-A Deoxy taxols BRISTOL MYERS SQUIBB CO (US) 1994-04-20 CN disclosed
CN-1082541-A Fluoro taxols BRISTOL MYERS SQUIBB CO (US) 1994-02-23 CN disclosed
CN-1069028-A The asymmetric synthesis of taxol side chain BRISTOL MYERS SQUIBB CO (US) 1993-02-17 CN disclosed