SCHEMBL27368748

SCHEMBL27368748

NCc1ccc([C@@H](C(=O)O)C2CCCC2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BDKRB2 P30411 1/20 0.48
ALOX5 P09917 2/20 0.45
HDAC6 Q9UBN7 1/20 0.45
EPHX1 P07099 2/20 0.45
HTR1E P28566 2/20 0.44
S1PR3 Q99500 2/20 0.44
MEN1 O00255 2/20 0.44
LMNA P02545 2/20 0.44
KMT2A Q03164 2/20 0.44
MAPT P10636 1/20 0.44
CHRM3 P20309 5/20 0.42
MITF O75030 1/20 0.39
CHRM2 P08172 1/20 0.39
HTR1A P08908 1/20 0.39
ADRA2A P08913 1/20 0.39
CHRM1 P11229 1/20 0.39
DRD1 P21728 1/20 0.39
SLC6A2 P23975 1/20 0.39
ADRA1A P35348 1/20 0.39
OPRM1 P35372 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27361339 1.00 BDKRB2 (0.48) BDKRB2ALOX5HDAC6EPHX1HTR1E
SCHEMBL10006210 0.84 NPC1 (0.46) ALOX5HDAC6EPHX1HTR1ES1PR3
SCHEMBL7013582 0.84 ALOX5 (0.45) ALOX5HDAC6EPHX1HTR1ES1PR3
SCHEMBL1069660 0.84 ALOX5 (0.45) ALOX5HDAC6EPHX1HTR1ES1PR3
SCHEMBL8634916 0.83 CHRM3 (0.47) ALOX5HDAC6EPHX1HTR1ES1PR3
SCHEMBL27372606 0.82 SLC6A3 (0.59) SLC6A2SLC6A3
SCHEMBL27388408 0.81 CHRM3 (0.46) ALOX5HDAC6EPHX1HTR1ES1PR3
SCHEMBL27483589 0.81 CHRM3 (0.46) ALOX5HDAC6EPHX1HTR1ES1PR3
SCHEMBL8636307 0.80 CHRM3 (0.49) ALOX5HDAC6EPHX1HTR1ES1PR3
SCHEMBL4242909 0.80 ALOX5 (0.49) ALOX5HDAC6HTR1ES1PR3MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102083803-B Oxocyclic substituted carboxylic acid derivatives and their use BAYER IP GMBH 2015-02-18 CN disclosed
CN-1330065-A Intermediates for the preparation of enantiomerically pure indole carboxylic acids and reactive derivatives thereof BAYER AG (DE) 2002-01-09 CN disclosed
CN-1312246-A Process for preparing carboxylic acid BAYER AG (DE) 2001-09-12 CN disclosed
CN-1067394-C Process for the preparation of enantiomerically pure indole-carboxylic acids and their reactive derivatives BAYER AG (DE) 2001-06-20 CN disclosed
CN-1067393-C Novel pyrimido [1, 2-a ] indoles BAYER AG (DE) 2001-06-20 CN disclosed
CN-1184109-A Process for the preparation of enantiomerically pure cycloalkanolindoleindole-and azaindole-and pyrimido [1, 2-a ] -indole-carboxylic acids and active derivatives thereof BAYER AG (DE) 1998-06-10 CN disclosed