SCHEMBL27375508

SCHEMBL27375508

CCC(=O)Oc1c(-c2ccc(F)cc2)c2ccsc2c(=O)n1C

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CENPE Q02224 4/20 0.35
PKM P14618 1/20 0.35
PKLR P30613 1/20 0.35
RXFP1 Q9HBX9 4/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.33
TACR1 P25103 1/20 0.33
GRIA2 P42262 1/20 0.33
GRIA4 P48058 1/20 0.33
NEK1 Q96PY6 2/20 0.32
MAPK14 Q16539 1/20 0.32
TP53 P04637 1/20 0.32
HTT P42858 1/20 0.32
PTGS1 P23219 1/20 0.32
PTGS2 P35354 1/20 0.32
DPP4 P27487 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27539886 0.89 ADORA3 (0.41) PKMTACR1TP53HTT
SCHEMBL27371705 0.82 CENPE (0.48) CENPETACR1GRIA2GRIA4MAPK14
SCHEMBL27399207 0.79 PKM (0.35) CENPEPKMPKLRRXFP1NEK1
SCHEMBL27364098 0.79 TP53 (0.35) CENPETACR1GRIA2GRIA4MAPK14
SCHEMBL7852329 0.78 TP53 (0.41) CENPEPKMTP53HTT
SCHEMBL27530229 0.77 GAA (0.34) PKMPKLRRXFP1TACR1TP53
SCHEMBL7850622 0.76 GRIA2 (0.44) CENPEPKMPKLRRXFP1TACR1
SCHEMBL7849856 0.70 TACR1 (0.66) RXFP1TACR1TP53HTT
SCHEMBL27364100 0.70 PKM (0.35) CENPEPKMPKLRTACR1NEK1
SCHEMBL7850615 0.69 GRIA2 (0.44) CENPEPKMPKLRTACR1GRIA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1052004-C Heterocyclic compounds, their production and use TALCEDA CHEMICAL IND LTD (JP) 2000-05-03 CN disclosed
CN-1107476-A Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1995-08-30 CN disclosed