SCHEMBL27397133

SCHEMBL27397133

COc1ccccc1N(C)C(=O)C(Cl)C(CCO)c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
CRHBP P24387 1/20 0.43
CRHR2 Q13324 1/20 0.43
L3MBTL1 Q9Y468 2/20 0.42
SLC6A2 P23975 1/20 0.40
SLC6A4 P31645 1/20 0.40
MAPK1 P28482 1/20 0.40
KCNA3 P22001 1/20 0.39
ALDH1A1 P00352 2/20 0.39
SLC6A9 P48067 1/20 0.38
TSPO P30536 1/20 0.36
HPGD P15428 1/20 0.36
POLB P06746 1/20 0.36
HTT P42858 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
PAX8 Q06710 1/20 0.36
TLR9 Q9NR96 1/20 0.36
GPBAR1 Q8TDU6 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27415579 0.81 MEN1 (0.65) MEN1KMT2ACRHBPCRHR2ALDH1A1
SCHEMBL27416258 0.81 LMNA (0.43) MEN1KMT2AL3MBTL1SLC6A2SLC6A4
SCHEMBL27398401 0.80 LMNA (0.36) SLC6A2SLC6A4ALDH1A1HPGD
SCHEMBL27430310 0.77 DRD4 (0.43) MEN1KMT2AL3MBTL1SLC6A2SLC6A4
SCHEMBL27396374 0.74 ACHE (0.47) MEN1KMT2ACRHBPCRHR2ALDH1A1
SCHEMBL28399460 0.72 TSPO (0.46) MEN1KMT2ACRHBPCRHR2L3MBTL1
SCHEMBL7811272 0.72 CDK8 (0.40) MEN1KMT2AALDH1A1GPBAR1
SCHEMBL27416257 0.72 MEN1 (0.49) MEN1KMT2AALDH1A1HPGDPOLB
SCHEMBL27415578 0.72 MLYCD (0.45) MEN1KMT2A
SCHEMBL20264683 0.71 ALDH1A1 (0.51) MEN1KMT2ACRHBPCRHR2L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1085661-C Piperidine derivatives as neurokinin antagonists SCHERING CORP (US) 2002-05-29 CN disclosed
CN-1161033-A Piperidine derivatives as neurokinin antagonists SCHERING CORP (US) 1997-10-01 CN disclosed