SCHEMBL27403138

SCHEMBL27403138

NC(=O)C1CN(C(c2ccccc2)c2ccccc2)CCN1C(=O)c1cccnc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1A O00555 2/20 0.49
CACNA2D1 P54289 2/20 0.49
CACNB1 Q02641 2/20 0.49
CACNA1C Q13936 1/20 0.49
MAOB P27338 1/20 0.44
PIK3CD O00329 1/20 0.44
NAMPT P43490 1/20 0.43
HPGD P15428 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
VNN1 O95497 1/20 0.42
LMNA P02545 1/20 0.42
ALDH1A1 P00352 1/20 0.41
HTT P42858 1/20 0.41
OPRM1 P35372 1/20 0.41
OPRD1 P41143 1/20 0.41
OPRK1 P41145 1/20 0.41
OPRL1 P41146 1/20 0.41
CHRNB2 P17787 1/20 0.40
CHRNB4 P30926 1/20 0.40
CHRNA3 P32297 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27403084 0.92 CACNA1A (0.58) CACNA1ACACNA2D1CACNB1CACNA1CMAOB
SCHEMBL27403135 0.86 CACNA1A (0.49) CACNA1ACACNA2D1CACNB1CACNA1CMAOB
SCHEMBL27402018 0.84 CACNA1A (0.44) CACNA1ACACNA2D1CACNB1CACNA1CMAOB
SCHEMBL27403139 0.82 MGLL (0.43) CACNA1ACACNA2D1CACNB1CACNA1CMAOB
SCHEMBL27403172 0.79 OPRD1 (0.45) CACNA1ACACNA2D1CACNB1CACNA1CMAOB
SCHEMBL27411313 0.77 PIK3CD (0.43) CACNA1ACACNA2D1CACNB1CACNA1CMAOB
SCHEMBL27411332 0.76 CYP1A2 (0.40) CACNA1ACACNA2D1CACNB1CACNA1CPIK3CD
SCHEMBL31350612 0.76 MAOB (0.70) MAOBNAMPTNPSR1OPRM1OPRD1
SCHEMBL5268550 0.75 CACNA2D1 (0.80) CACNA1ACACNA2D1CACNB1CACNA1C
SCHEMBL31350763 0.74 L3MBTL1 (0.46) MAOBPIK3CDNAMPTLMNAOPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024124287-A1 COMPOUNDS FOR TREATING VIRAL INFECTION THE WALTER AND ELIZA HALL INSTITUTE OF MEDICAL RESEARCH (AU) 2024-06-20 WO disclosed