SCHEMBL27410085

SCHEMBL27410085

CCCNN1CCN(c2cccc3ccccc23)CC1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 5/20 0.50
HTR2A P28223 3/20 0.50
HTR7 P34969 3/20 0.50
HTR3A P46098 2/20 0.50
HTR3E A5X5Y0 1/20 0.50
HTR3B O95264 1/20 0.50
CYP1A2 P05177 1/20 0.50
CYP2D6 P10635 1/20 0.50
NCF1 P14598 1/20 0.50
TSHR P16473 1/20 0.50
NFKB1 P19838 1/20 0.50
HTR1D P28221 1/20 0.50
HTR1B P28222 1/20 0.50
MTOR P42345 1/20 0.50
HTR5A P47898 1/20 0.50
HTR6 P50406 1/20 0.50
HTR3D Q70Z44 1/20 0.50
HTR3C Q8WXA8 1/20 0.50
HSD17B10 Q99714 1/20 0.50
SIGMAR1 Q99720 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8828451 0.80 DRD2 (0.45) HTR1AHTR2ANCF1TSHRHSD17B10
SCHEMBL8828572 0.80 ADRB1 (0.49) HTR7TSHRHSD17B10ALDH1A1LMNA
SCHEMBL8828393 0.79 HSD17B10 (0.55) TSHRNFKB1HSD17B10KDM4EALDH1A1
SCHEMBL9643856 0.79 HTR1A (0.74) HTR1AHTR2AHTR7HTR3AHTR3E
SCHEMBL4249373 0.78 TSHR (0.56) TSHRHSD17B10KDM4EALDH1A1LMNA
SCHEMBL8828348 0.78 BRD9 (0.40) HTR1AHTR2ANCF1KDM4EALDH1A1
Hydrochloric Acid SCHEMBL7203515 0.77 KDM4E (0.75) HTR1AHTR2AHTR7HTR3AHTR3E
SCHEMBL8828453 0.77 DRD4 (0.46) HTR1AHTR2AHTR7CYP1A2CYP2D6
SCHEMBL8828510 0.77 DRD2 (0.62) HTR1AHTR3AHTR3EHTR3BCYP1A2
SCHEMBL8828437 0.77 HTR1A (0.41) HTR1AHTR7TSHRDRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1074766-C Alkylaminobenzothiazole and -benzoxazole derivatives JANSSEN PHARMACEUTICA NV (BE) 2001-11-14 CN disclosed
CN-1218461-A Alkylaminobenzothiazole and -benzoxazole derivatives JANSSEN PHARMACEUTICA NV (NL) 1999-06-02 CN disclosed