SCHEMBL27410461

SCHEMBL27410461

CCOC(=O)c1nnc(-c2cccnc2)n1-c1c(Cl)ccc2nc(OC)c(OC)nc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 3/20 0.41
HTT P42858 2/20 0.40
ALDH1A1 P00352 4/20 0.40
TSHR P16473 2/20 0.40
GAA P10253 1/20 0.40
DCTPP1 Q9H773 1/20 0.40
LMNA P02545 1/20 0.39
POLB P06746 1/20 0.39
KDM4E B2RXH2 2/20 0.39
PDE2A O00408 1/20 0.39
APLNR P35414 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
MAPT P10636 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
MMP2 P08253 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27434412 0.91 PDE2A (0.44) HTTALDH1A1LMNAPOLBPDE2A
SCHEMBL7676180 0.90 ACHE (0.40) ACHEHTTALDH1A1TSHRGAA
SCHEMBL27433674 0.84 MAPT (0.36) HTTALDH1A1GAAPOLBKDM4E
SCHEMBL27489462 0.83 APLNR (0.41) HTTALDH1A1TSHRPDE2AAPLNR
SCHEMBL27502563 0.82 APLNR (0.43) HTTALDH1A1PDE2AAPLNRMAPK1
SCHEMBL27541050 0.81 APLNR (0.41) HTTALDH1A1PDE2AAPLNRMAPT
SCHEMBL7682502 0.80 PDE2A (0.43) HTTALDH1A1TSHRLMNAPOLB
SCHEMBL27409634 0.75 PDE10A (0.37) HTTALDH1A1GAAKDM4EPDE2A
SCHEMBL27435510 0.75 DYRK1A (0.35) HTTALDH1A1GAAPOLBKDM4E
SCHEMBL27487153 0.72 GLA (0.37) ALDH1A1APLNRMAPTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1103770-C Quinoxalinediones PFIZER RES AND DEV CO N V S A (IE) 2003-03-26 CN disclosed
CN-1213369-A Quinoxalinedione compound PFIZER RES & DEV (IE) 1999-04-07 CN disclosed