SCHEMBL27430682

SCHEMBL27430682

[O]C1(c2cccc(O)c2)CCCC1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRD1 P41143 3/20 0.46
OPRM1 P35372 5/20 0.44
SLC6A4 P31645 3/20 0.44
ACHE P22303 2/20 0.44
SLC22A1 O15245 1/20 0.44
CHRM2 P08172 1/20 0.44
CYP2D6 P10635 1/20 0.44
SLC6A2 P23975 2/20 0.43
OPRK1 P41145 2/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
CA12 O43570 1/20 0.42
ALDH1A1 P00352 1/20 0.42
CA2 P00918 1/20 0.42
LMNA P02545 1/20 0.42
CYP3A4 P08684 1/20 0.42
CA5A P35218 1/20 0.42
CA9 Q16790 1/20 0.42
HSD17B10 Q99714 1/20 0.42
CA14 Q9ULX7 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30475863 0.78 ESR1 (0.57) OPRD1OPRM1SLC6A4ACHESLC22A1
SCHEMBL3946783 0.76 OPRM1 (0.47) OPRD1OPRM1SLC6A4ACHESLC22A1
SCHEMBL14531297 0.76 AKR1C1 (0.67) CYP2D6MEN1KMT2A
SCHEMBL5808986 0.74 OPRD1 (0.67) OPRD1OPRM1SLC6A4ACHESLC22A1
SCHEMBL7802441 0.74 LMNA (0.53) OPRD1LMNA
SCHEMBL6417291 0.74 AKR1C1 (0.65) CYP2D6MEN1KMT2A
SCHEMBL12020311 0.74 HDAC4 (0.49) OPRD1OPRM1SLC6A4ACHESLC22A1
SCHEMBL19646503 0.73 ESR1 (0.57) OPRD1OPRM1ACHEOPRK1ALDH1A1
SCHEMBL27906398 0.72 SLC6A4 (0.50) SLC6A4SLC6A2MEN1KMT2AALDH1A1
SCHEMBL15021523 0.72 OPRD1 (0.46) OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1109683-C 2-arylbenzo [ b ] thiophenes for the treatment of estrogen deficiency syndrome LILLY CO ELI (US) 2003-05-28 CN claimed
CN-1278811-A 2-arylbenzo [ b ] thiophenes for the treatment of estrogen deficiency syndrome LILLY CO ELI (US) 2001-01-03 CN claimed
CN-1109683-C 2-arylbenzo [ b ] thiophenes for the treatment of estrogen deficiency syndrome LILLY CO ELI (US) 2003-05-28 CN disclosed
CN-1278811-A 2-arylbenzo [ b ] thiophenes for the treatment of estrogen deficiency syndrome LILLY CO ELI (US) 2001-01-03 CN disclosed