SCHEMBL27433853

SCHEMBL27433853

C[CH]CN1CCN(c2ccccc2C2CC2)CC1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.48
ADRA1B P35368 1/20 0.48
KDM4E B2RXH2 3/20 0.43
TDP1 Q9NUW8 1/20 0.43
GAA P10253 1/20 0.40
HPGD P15428 1/20 0.40
ALDH1A1 P00352 1/20 0.39
PLA2G1B P04054 1/20 0.39
RAB9A P51151 1/20 0.39
ATG4B Q9Y4P1 1/20 0.39
SLC6A2 P23975 1/20 0.39
SLC6A4 P31645 1/20 0.39
DRD4 P21917 1/20 0.39
DRD3 P35462 1/20 0.39
LMNA P02545 1/20 0.38
MAPT P10636 1/20 0.38
SIGMAR1 Q99720 1/20 0.37
HTR2C P28335 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9853259 0.79 CARM1 (0.55) HTR1AADRA1BSIGMAR1
Hydrochloric Acid SCHEMBL9739959 0.78 CARM1 (0.54) HTR1AADRA1BSIGMAR1
SCHEMBL8297825 0.77 HTR1A (0.50) HTR1AADRA1BKDM4ESLC6A2SLC6A4
SCHEMBL23064518 0.77 ADRA2C (0.55) HTR1AADRA1BKDM4EHPGDALDH1A1
SCHEMBL27597994 0.76 DRD2 (0.48) HTR1AKDM4ETDP1ALDH1A1PLA2G1B
SCHEMBL27597996 0.76 KDM4E (0.66) KDM4ETDP1GAAALDH1A1DRD4
Hydrochloric Acid SCHEMBL9134644 0.76 HTR1A (0.49) HTR1AADRA1BKDM4ESLC6A2SLC6A4
SCHEMBL8828503 0.75 CYP2D6 (0.56) HTR1AADRA1BKDM4ESLC6A4LMNA
SCHEMBL31198346 0.75 KEAP1 (0.48) HTR1AADRA1BKDM4EGAAALDH1A1
SCHEMBL23064483 0.75 KEAP1 (0.48) HTR1AADRA1BKDM4EGAAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1104637-A Derivative of 2-aminopyrazine-5-carboxamide, preparation and pharmaceutical use of same SYNTHELABO (FR) 1995-07-05 CN disclosed