SCHEMBL2745009

SCHEMBL2745009

COc1cc(-c2ccc[c]n2)ccc1OCCN1CCC(N(C)C)CC1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 1/20 0.48
NOS1 P29475 1/20 0.48
NOS2 P35228 1/20 0.48
MCHR1 Q99705 3/20 0.43
ADRA1A P35348 2/20 0.41
ADRA1B P35368 2/20 0.41
MAP3K11 Q16584 2/20 0.41
LTA4H P09960 1/20 0.40
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.39
ALDH1A1 P00352 1/20 0.39
KMT2A Q03164 1/20 0.39
HRH3 Q9Y5N1 2/20 0.39
GRM4 Q14833 1/20 0.39
ABL1 P00519 1/20 0.38
KIT P10721 1/20 0.38
SRC P12931 1/20 0.38
FRK P42685 1/20 0.38
PTK6 Q13882 1/20 0.38
ADORA2A P29274 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27981872 0.87 LTA4H (0.53) MCHR1LTA4HHRH3ADORA2AADORA1
SCHEMBL221350 0.83 NOS1 (0.67) NOS3NOS1NOS2MCHR1ADRA1A
SCHEMBL27981880 0.78 NOS3 (0.46) NOS3NOS1NOS2MCHR1KDM4E
SCHEMBL5538401 0.73 KDM4E (0.49) KDM4EMEN1ALDH1A1KMT2A
SCHEMBL4741439 0.69 ROCK2 (0.40) NOS3NOS1NOS2KDM4EMEN1
SCHEMBL220877 0.68 NOS3 (0.61) NOS3NOS1NOS2MCHR1LTA4H
SCHEMBL219485 0.68 NOS3 (0.64) NOS3NOS1NOS2MCHR1
SCHEMBL27981548 0.68 PTPN1 (0.48) LTA4HKDM4EALDH1A1HRH3
SCHEMBL6957842 0.66 MCHR1 (0.70) MCHR1LTA4HHTR2A
SCHEMBL6847455 0.66 HRH3 (0.80) HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8178536-B2 Sirtuin modulating compounds SIRTRIS PHARMACEUTICALS, INC. (US) 2012-05-15 US disclosed