SCHEMBL27465652

SCHEMBL27465652

CS(=O)(=O)c1cc(C[O])cc(-c2ccc(F)cc2)c1

nearest known ligand 0.50

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.50
LOX P28300 1/20 0.50
PTGS2 P35354 17/20 0.49
LOXL2 Q9Y4K0 2/20 0.47
PTGS1 P23219 3/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27466225 0.86 MAOA (0.49) MAOALOXPTGS2LOXL2PTGS1
SCHEMBL7395459 0.74 PTGS2 (0.74) PTGS2PTGS1
SCHEMBL6470141 0.74 PTGS2 (0.74) PTGS2PTGS1
SCHEMBL5831675 0.73 PTGS2 (0.56) MAOAPTGS2PTGS1
SCHEMBL27709191 0.70 MAOB (0.52) LOXL2
SCHEMBL27431456 0.70 PTPN5 (0.54) PTGS2PTGS1
SCHEMBL5898253 0.70 PTGS2 (0.37) LOXPTGS2LOXL2PTGS1
SCHEMBL444872 0.68 PTGS2 (0.69) PTGS2PTGS1
SCHEMBL7935589 0.66 PTGS2 (0.56) PTGS2PTGS1
SCHEMBL7054313 0.66 ALDH1A1 (0.47) LOXLOXL2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1155600-C 2, 3-diaryl pyrazolo [1, 5-b ] pyridazine derivatives, their preparation and their use as cyclooxygenase 2 inhibitors 2004-06-30 CN disclosed
CN-1278263-A 2,3-diaryl-pyrazolo [1,5-B] pyridazines derivatives, their prepn. and use as cyclooxygenase 2 (cox-2) inhibitors GLAXO GROUP LTD (GB) 2000-12-27 CN disclosed