SCHEMBL2748265

SCHEMBL2748265

FC(F)(F)c1cccc2sc(S)nc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
AKR1B1 P15121 1/20 0.38
MPL P40238 3/20 0.37
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
GAA P10253 3/20 0.35
KDM4E B2RXH2 1/20 0.35
LMNA P02545 1/20 0.35
PRNP P04156 1/20 0.35
HPGD P15428 1/20 0.35
PARP1 P09874 1/20 0.35
MAPT P10636 2/20 0.33
SLC9A1 P19634 1/20 0.33
HDAC3 O15379 1/20 0.33
HDAC4 P56524 1/20 0.33
HDAC1 Q13547 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24818889 0.80 ALDH1A1 (0.40) ALDH1A1L3MBTL1AKR1B1MPLMEN1
SCHEMBL22891113 0.80 ALDH1A1 (0.43) ALDH1A1L3MBTL1AKR1B1MPLMEN1
SCHEMBL3067465 0.79 PSMD14 (0.42) ALDH1A1L3MBTL1MEN1KMT2ANPC1
SCHEMBL1913695 0.79 ALDH1A1 (0.61) ALDH1A1L3MBTL1AKR1B1MPLMEN1
SCHEMBL2747730 0.79 ALDH1A1 (0.56) ALDH1A1L3MBTL1AKR1B1MPLMEN1
SCHEMBL25367519 0.79 ALDH1A1 (0.39) ALDH1A1L3MBTL1AKR1B1MPLMEN1
SCHEMBL8977752 0.77 AKR1B1 (0.40) ALDH1A1L3MBTL1AKR1B1MPLMEN1
SCHEMBL2252871 0.77 PSMD14 (0.41) ALDH1A1L3MBTL1MEN1KMT2ANPC1
SCHEMBL2256808 0.77 PSMD14 (0.41) ALDH1A1L3MBTL1MEN1KMT2ANPC1
Hydrogen Sulfide SCHEMBL27391083 0.77 ALDH1A1 (0.32) ALDH1A1MEN1KMT2AGAAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12577240-B2 Antiviral heteroaryl ketone derivatives PFIZER INC. (US) 2026-03-17 US disclosed
US-20230339930-A1 Antiviral Heteroaryl Ketone Derivatives PFIZER INC. (US) 2023-10-26 US disclosed
US-20230339930-A1 Antiviral Heteroaryl Ketone Derivatives PFIZER INC. (US) 2023-10-26 US disclosed
US-20230339930-A1 Antiviral Heteroaryl Ketone Derivatives PFIZER INC. (US) 2023-10-26 US disclosed
EP-4178955-A1 ANTIVIRAL HETEROARYL KETONE DERIVATIVES Pfizer Inc. (US) 2023-05-17 EP disclosed
WO-2022013684-A1 ANTIVIRAL HETEROARYL KETONE DERIVATIVES PFIZER INC. (US) 2022-01-20 WO disclosed
WO-2022013684-A1 ANTIVIRAL HETEROARYL KETONE DERIVATIVES PFIZER INC. (US) 2022-01-20 WO disclosed
CN-104478828-A 2-amino-7-substituted benzothiazole compound as well as preparation method and application thereof ZHANGZHOU PIEN TZE HUANG PHARM 2015-04-01 CN disclosed
US-8178668-B2 2-aminopyridine kinase inhibitors OSI Pharmaceuticals, LLC (US) 2012-05-15 US disclosed
EP-2265270-A1 2-AMINOPYRIDINE KINASE INHIBITORS OSI Pharmaceuticals, Inc. (US) 2010-12-29 EP disclosed
WO-2009099982-A1 2-AMINOPYRIDINE KINASE INHIBITORS OSI PHARMACEUTICALS, INC. (US) 2009-08-13 WO disclosed
US-20090197862-A1 2-AMINOPYRIDINE KINASE INHIBITORS OSI PHARMACEUTICALS, INC. 2009-08-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12577240-B2 Antiviral heteroaryl ketone derivatives ACE2, SARS1, ACE ALDH1A1 1752/4885L3MBTL1 1241/4885AKR1B1 785/4885
US-20230339930-A1 Antiviral Heteroaryl Ketone Derivatives ACE2, ZC3HAV1, SARS1 ALDH1A1 1519/4885L3MBTL1 489/4885AKR1B1 197/4885
US-20090197862-A1 2-AMINOPYRIDINE KINASE INHIBITORS ERBB2, ABL2, TIE1 ALDH1A1 945/4885L3MBTL1 3088/4885AKR1B1 716/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.