SCHEMBL28200415

SCHEMBL28200415

COC(=O)CC(C)Cc1ccc(F)cc1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.49
ALDH1A1 P00352 1/20 0.49
MAPT P10636 1/20 0.49
HPGD P15428 1/20 0.47
TRPA1 O75762 1/20 0.46
TSHR P16473 1/20 0.46
CA12 O43570 3/20 0.44
CA7 P43166 3/20 0.44
CA9 Q16790 3/20 0.44
CA14 Q9ULX7 3/20 0.44
CA2 P00918 1/20 0.44
NOS3 P29474 1/20 0.44
NOS1 P29475 1/20 0.44
NOS2 P35228 1/20 0.44
KMT2A Q03164 3/20 0.43
MEN1 O00255 2/20 0.43
GAA P10253 1/20 0.43
KLK7 P49862 1/20 0.42
TDP1 Q9NUW8 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27488012 0.85 HTT (0.43) HTTALDH1A1MAPTHPGDTRPA1
SCHEMBL25832024 0.85 ACACB (0.44) ALDH1A1HPGDKMT2AMEN1TDP1
SCHEMBL19479754 0.85 ESR1 (0.53) MAPTTSHRKMT2AGAA
SCHEMBL7710947 0.85 ESR1 (0.53) MAPTTSHRKMT2AGAA
SCHEMBL13610016 0.84 KMT2A (0.47) HTTALDH1A1MAPTHPGDTSHR
SCHEMBL13643084 0.83 F2 (0.43) ALDH1A1MAPTGAA
SCHEMBL22769201 0.83 RAB9A (0.54) ALDH1A1MAPTHPGDTSHRKMT2A
SCHEMBL10509525 0.83 NPC1 (0.51) ALDH1A1TSHRKMT2AMEN1
SCHEMBL27506588 0.81 CA12 (0.47) HTTALDH1A1MAPTHPGDTRPA1
SCHEMBL5794436 0.81 TRPA1 (0.50) HTTHPGDTRPA1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108093636-A Indoleamine 2, 3-dioxygenase inhibitors for the treatment of cancer 百时美施贵宝公司 2018-05-29 CN disclosed
CN-107743481-A Indoleamine 2, 3-dioxygenase inhibitors for the treatment of cancer 百时美施贵宝公司 2018-02-27 CN disclosed
CN-107743490-A For the indoleamine 2 for the treatment of cancer, 3 dioxygenase inhibitors 百时美施贵宝公司 2018-02-27 CN disclosed