SCHEMBL27488605

SCHEMBL27488605

CC(C)CCc1c(-c2ccc(C[SH](=O)=O)cc2)cnn(-c2ccc(F)c(Cl)c2)c1=O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPBWR1 P48145 3/20 0.36
MCHR1 Q99705 1/20 0.36
ALDH1A1 P00352 3/20 0.35
ESR1 P03372 1/20 0.35
POLB P06746 1/20 0.35
HPGD P15428 1/20 0.35
IDO1 P14902 6/20 0.35
TDO2 P48775 6/20 0.35
CYP17A1 P05093 1/20 0.33
CYP1A2 P05177 1/20 0.33
GRM2 Q14416 1/20 0.33
KDM4E B2RXH2 1/20 0.33
TSHR P16473 1/20 0.33
MEN1 O00255 1/20 0.33
MAPT P10636 1/20 0.33
KMT2A Q03164 1/20 0.33
AVPR1B P47901 2/20 0.33
BRD9 Q9H8M2 1/20 0.32
TRPC5 Q9UL62 1/20 0.32
AR P10275 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27486810 0.88 RAB9A (0.42) NPBWR1MCHR1MAPTKMT2ATRPC5
SCHEMBL27470577 0.86 RAB9A (0.43) NPBWR1MCHR1ALDH1A1HPGDCYP1A2
SCHEMBL4191773 0.86 ALDH1A1 (0.35) ALDH1A1ESR1POLBHPGDIDO1
SCHEMBL4189784 0.85 PTGS2 (0.46) IDO1TDO2
SCHEMBL4186306 0.84 PTGS2 (0.45)
SCHEMBL27487528 0.84 SMN1; SMN2 (0.38) NPBWR1MCHR1ALDH1A1ESR1POLB
SCHEMBL27471545 0.83 IDO1 (0.38) NPBWR1MCHR1ALDH1A1ESR1POLB
SCHEMBL27549347 0.82 RAB9A (0.40) NPBWR1MCHR1MAPTKMT2ATRPC5
SCHEMBL4180594 0.82 AR (0.36) ALDH1A1ESR1POLBHPGDIDO1
SCHEMBL27555435 0.81 RAB9A (0.41) NPBWR1MCHR1ALDH1A1HPGDCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1167687-C Arylpyridazinones as prostaglandin endoperoxide H synthase biosynthesis inhibitors ���Ͽع����޹�˾ 2004-09-22 CN disclosed
CN-1277605-A Arylpyridazinones as prostaglandin endoperoxide H synthase biosynthesis inhibitors ABBOTT LAB (US) 2000-12-20 CN disclosed