SCHEMBL27490983

SCHEMBL27490983

O=COCCc1c(-c2ccncc2)c(-c2cccs2)n2c1CCC2

nearest known ligand 0.36

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 2/20 0.36
KCNH2 Q12809 1/20 0.31
HRH3 Q9Y5N1 1/20 0.31
SIGMAR1 Q99720 1/20 0.31
PTGS1 P23219 1/20 0.30
CYP17A1 P05093 1/20 0.30
CYP11B1 P15538 1/20 0.30
CYP11B2 P19099 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27491679 0.85 PTGS1 (0.36) PTGS1
SCHEMBL27511308 0.82 KMT2A (0.41)
SCHEMBL27509845 0.82 KMT2A (0.41)
SCHEMBL6290812 0.74 KMT2A (0.44) ALOX5
SCHEMBL7006701 0.73 ALOX5 (0.41) ALOX5
SCHEMBL6294039 0.72 ALDH1A1 (0.47)
SCHEMBL7006366 0.71 KMT2A (0.38) ALOX5
SCHEMBL6294501 0.71 KCNK3 (0.48)
Ethoxycarbonyl Group SCHEMBL27490984 0.71 GABRA1 (0.39)
SCHEMBL7013150 0.69 KMT2A (0.40) ALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1206230-C 4-Pyridyl-and 2,4-pyrimidinyl-substituted pyrrole derivatives and their use in pharmacy MERCKLE GMBH (DE) 2005-06-15 CN disclosed
CN-1396923-A 4-Pyridyl-and 2,4-pyrimidinyl-substituted pyrrole derivatives and their use in pharmacy MERCKLE GMBH (DE) 2003-02-12 CN disclosed