SCHEMBL27501985

SCHEMBL27501985

NN=CNc1cccc(C(=O)NCC(=O)NCC(C(=O)O)c2ccccc2)c1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 5/20 0.44
ITGA5 P08648 5/20 0.44
ITGB3 P05106 4/20 0.44
ITGAV P06756 4/20 0.44
MDM4 O15151 2/20 0.44
GPR139 Q6DWJ6 10/20 0.42
MDM2 Q00987 2/20 0.42
NPC1 O15118 1/20 0.41
KMT2A Q03164 2/20 0.41
MEN1 O00255 1/20 0.41
ATM Q13315 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.38
TAAR1 Q96RJ0 1/20 0.38
HTT P42858 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27486185 0.89 ALDH1A1 (0.41) ITGB1ITGA5ITGB3ITGAVMDM4
SCHEMBL27503083 0.89 HTT (0.43) ITGB1ITGA5ITGB3ITGAVMDM4
SCHEMBL27486186 0.89 ITGB1 (0.39) ITGB1ITGA5ITGB3ITGAVMDM4
SCHEMBL27486190 0.88 GPR139 (0.46) ITGB1ITGA5GPR139KMT2AMEN1
SCHEMBL27521095 0.86 KMT2A (0.42) ITGB1ITGA5GPR139NPC1KMT2A
SCHEMBL27484439 0.85 ITGB1 (0.39) ITGB1ITGA5ITGB3ITGAVMDM4
SCHEMBL27504167 0.85 ITGB1 (0.51) ITGB1ITGA5ITGB3ITGAVMDM4
SCHEMBL242675 0.83 ITGB1 (0.45) ITGB1ITGA5ITGB3ITGAVMDM4
SCHEMBL27522236 0.83 ITGB1 (0.41) ITGB1ITGA5ITGB3ITGAVGPR139
SCHEMBL27555002 0.83 HTT (0.43) ITGB1ITGA5ITGB3ITGAVNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1201454-A Meta-guanidino, ureido, thioureido or azacyclic aminobenzoic acid derivatives as integrin antagonists SEARLE & CO (US) 1998-12-09 CN claimed