SCHEMBL27484439

SCHEMBL27484439

NN=CNc1cccc(C(=O)NCC(=O)NCC(C(=O)O)c2ccccc2OCC(=O)O)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 3/20 0.39
ITGA5 P08648 3/20 0.39
KMT2A Q03164 3/20 0.39
PKM P14618 1/20 0.39
HTT P42858 1/20 0.39
MAPK1 P28482 1/20 0.38
GPR139 Q6DWJ6 2/20 0.38
MEN1 O00255 2/20 0.37
POLB P06746 2/20 0.37
ITGB3 P05106 3/20 0.36
ITGAV P06756 2/20 0.36
MDM4 O15151 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
ITGA2B P08514 1/20 0.36
KDM4E B2RXH2 1/20 0.36
NPC1 O15118 1/20 0.35
MITF O75030 1/20 0.35
NFKB1 P19838 1/20 0.35
RAB9A P51151 1/20 0.35
NFKB2 Q00653 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27502752 0.91 KMT2A (0.41) ITGB1ITGA5KMT2APKMHTT
SCHEMBL27501985 0.85 ITGB1 (0.44) ITGB1ITGA5KMT2AHTTGPR139
SCHEMBL27503083 0.84 HTT (0.43) ITGB1ITGA5KMT2APKMHTT
SCHEMBL6777703 0.84 ITGB3 (0.46) ITGB1ITGA5ITGB3ITGAVMDM4
SCHEMBL27521095 0.82 KMT2A (0.42) ITGB1ITGA5KMT2AMAPK1GPR139
SCHEMBL7340359 0.81 GPR139 (0.40) ITGB1ITGA5KMT2APKMHTT
SCHEMBL27522236 0.81 ITGB1 (0.41) ITGB1ITGA5KMT2AGPR139MEN1
SCHEMBL27555002 0.81 HTT (0.43) ITGB1ITGA5KMT2AHTTMAPK1
SCHEMBL27486190 0.80 GPR139 (0.46) ITGB1ITGA5KMT2APKMHTT
SCHEMBL27503085 0.79 ITGB3 (0.47) ITGB1ITGA5KMT2AHTTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1201454-A Meta-guanidino, ureido, thioureido or azacyclic aminobenzoic acid derivatives as integrin antagonists SEARLE & CO (US) 1998-12-09 CN claimed