SCHEMBL27555002

SCHEMBL27555002

NN=CNc1cccc(C(=O)NCC(=O)NCC(C(=O)O)c2cc(Br)ccc2O)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 4/20 0.43
LMNA P02545 3/20 0.43
KDM4E B2RXH2 2/20 0.43
MAPT P10636 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
ITGB3 P05106 6/20 0.38
ITGAV P06756 6/20 0.38
ITGB6 P18564 6/20 0.38
ITGB1 P05556 2/20 0.38
ITGA5 P08648 2/20 0.38
ITGB5 P18084 1/20 0.38
ITGB8 P26012 1/20 0.38
ITGA8 P53708 1/20 0.38
NPC1 O15118 1/20 0.38
GAA P10253 1/20 0.38
RAB9A P51151 1/20 0.38
MEN1 O00255 1/20 0.37
MAPK1 P28482 1/20 0.37
KMT2A Q03164 1/20 0.37
TDP1 Q9NUW8 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27522236 0.90 ITGB1 (0.41) KDM4EITGB3ITGAVITGB6ITGB1
SCHEMBL27484813 0.87 ITGB3 (0.47) HTTLMNAKDM4EMAPTITGB3
SCHEMBL7345759 0.84 ITGB3 (0.56) HTTLMNAKDM4EMAPTSMN1; SMN2
SCHEMBL27503085 0.84 ITGB3 (0.47) HTTLMNAKDM4EMAPTITGB3
SCHEMBL27501985 0.83 ITGB1 (0.44) HTTSMN1; SMN2ITGB3ITGAVITGB1
SCHEMBL7345869 0.81 HTT (0.43) HTTLMNAKDM4EMAPTSMN1; SMN2
SCHEMBL27484439 0.81 ITGB1 (0.39) HTTKDM4ESMN1; SMN2ITGB3ITGAV
SCHEMBL27521095 0.78 KMT2A (0.42) LMNAMAPTSMN1; SMN2ITGB1ITGA5
SCHEMBL27486190 0.78 GPR139 (0.46) HTTKDM4ESMN1; SMN2ITGB1ITGA5
SCHEMBL27486185 0.77 ALDH1A1 (0.41) ITGB3ITGAVITGB1ITGA5NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1201454-A Meta-guanidino, ureido, thioureido or azacyclic aminobenzoic acid derivatives as integrin antagonists SEARLE & CO (US) 1998-12-09 CN claimed