SCHEMBL27520124

SCHEMBL27520124

CCCCOC(=O)c1ccnc(C(=O)O)c1N

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.52
HSD17B10 Q99714 3/20 0.52
TSHR P16473 6/20 0.51
L3MBTL1 Q9Y468 5/20 0.51
TDP1 Q9NUW8 2/20 0.51
LMNA P02545 6/20 0.48
CYP3A4 P08684 3/20 0.48
CYP1A2 P05177 2/20 0.48
CYP2C19 P33261 2/20 0.48
CYP2C9 P11712 1/20 0.48
PDE4D Q08499 1/20 0.48
MAPK1 P28482 3/20 0.47
KDM4E B2RXH2 2/20 0.47
POLB P06746 1/20 0.47
TP53 P04637 1/20 0.47
MAPT P10636 3/20 0.43
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
ESR1 P03372 1/20 0.42
CYP2D6 P10635 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15758316 0.77 NUDT1 (0.51) ALDH1A1HSD17B10TSHRLMNACYP3A4
SCHEMBL13133330 0.76 ALDH1A1 (0.64) ALDH1A1HSD17B10TSHRL3MBTL1TDP1
SCHEMBL13133331 0.76 ALDH1A1 (0.64) ALDH1A1HSD17B10TSHRL3MBTL1TDP1
SCHEMBL28182000 0.75 TSHR (0.48) ALDH1A1HSD17B10TSHRL3MBTL1TDP1
SCHEMBL8599944 0.74 ALDH1A1 (0.49) ALDH1A1HSD17B10TSHRL3MBTL1TDP1
SCHEMBL8405883 0.74 TSHR (0.66) ALDH1A1HSD17B10TSHRL3MBTL1TDP1
SCHEMBL7080700 0.74 KDM4E (0.42) ALDH1A1TSHRL3MBTL1TDP1LMNA
SCHEMBL9509719 0.74 LMNA (0.48) ALDH1A1HSD17B10TSHRL3MBTL1TDP1
SCHEMBL18159123 0.74 KDM4E (0.60) ALDH1A1TSHRL3MBTL1TDP1CYP3A4
SCHEMBL2595579 0.73 ALDH1A1 (0.64) ALDH1A1HSD17B10TSHRL3MBTL1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1226888-A Fluorinated 1,4-disubstituted piperidine derivatives BANYU PHARMA CO LTD (JP) 1999-08-25 CN disclosed