SCHEMBL2754552

SCHEMBL2754552

Brc1ccc(-c2cc(-c3cccc4ccccc34)nc(-c3ccccc3)n2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 1/20 0.50
CYP1A1 P04798 2/20 0.49
CYP1A2 P05177 2/20 0.49
CYP1B1 Q16678 2/20 0.49
MEN1 O00255 6/20 0.49
KMT2A Q03164 6/20 0.49
ALDH1A1 P00352 5/20 0.49
MAPT P10636 5/20 0.49
HPGD P15428 4/20 0.49
NTSR1 P30989 1/20 0.49
KDM4E B2RXH2 4/20 0.47
LMNA P02545 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
TP53 P04637 1/20 0.47
TSHR P16473 1/20 0.47
NFKB1 P19838 1/20 0.47
MAPK1 P28482 1/20 0.47
NFKB2 Q00653 1/20 0.47
RELA Q04206 1/20 0.47
ATM Q13315 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19383618 1.00 AGTR1 (0.50) AGTR1CYP1A1CYP1A2CYP1B1MEN1
SCHEMBL14416408 0.94 CYP1B1 (0.50) AGTR1CYP1A1CYP1A2CYP1B1MEN1
SCHEMBL15502106 0.93 AGTR1 (0.49) AGTR1CYP1A1CYP1A2CYP1B1MEN1
SCHEMBL19383283 0.91 AGTR1 (0.45) AGTR1CYP1A1CYP1A2CYP1B1MEN1
SCHEMBL10051210 0.91 MEN1 (0.54) CYP1A2MEN1KMT2AALDH1A1MAPT
SCHEMBL12306181 0.91 MEN1 (0.54) CYP1A2MEN1KMT2AALDH1A1MAPT
SCHEMBL10051196 0.91 MEN1 (0.54) CYP1A2MEN1KMT2AALDH1A1MAPT
SCHEMBL10051293 0.91 MEN1 (0.54) CYP1A2MEN1KMT2AALDH1A1MAPT
SCHEMBL14725231 0.91 MAPT (0.54) CYP1A2MEN1KMT2AALDH1A1MAPT
SCHEMBL17969997 0.89 MEN1 (0.53) MEN1KMT2AALDH1A1MAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20190106391-A1 COMPOUNDS WITH SPIROBIFLUORENE-STRUCTURES MERCK PATENT GMBH (DE) 2019-04-11 US disclosed
WO-2017157983-A1 COMPOUNDS WITH SPIROBIFLUORENE-STRUCTURES MERCK PATENT GMBH (DE) 2017-09-21 WO disclosed
US-9523031-B2 Organic electroluminescent device IDEMITSU KOSAN CO., LTD. (JP) 2016-12-20 US disclosed
US-9523031-B2 Organic electroluminescent device IDEMITSU KOSAN CO., LTD. (JP) 2016-12-20 US disclosed
US-20140018536-A1 AROMATIC AMINE DERIVATIVE AND ORGANIC ELECTROLUMINESCENCE DEVICE USING THE SAME IDEMITSU KOSAN CO., LTD. (JP) 2014-01-16 US disclosed
US-20140018536-A1 AROMATIC AMINE DERIVATIVE AND ORGANIC ELECTROLUMINESCENCE DEVICE USING THE SAME IDEMITSU KOSAN CO., LTD. (JP) 2014-01-16 US disclosed
US-8586206-B2 Aromatic amine derivative and organic electroluminescence device using the same IDEMITSU KOSAN CO., LTD. (JP) 2013-11-19 US disclosed
EP-2589596-A1 AROMATIC AMINE DERIVATIVE, AND ORGANIC ELECTROLUMINESCENT ELEMENT COMPRISING SAME Idemitsu Kosan Co., Ltd. (JP) 2013-05-08 EP disclosed
US-20120001154-A1 Aromatic amine derivative and organic electroluminescence device using the same IDEMITSU KOSAN CO., LTD. 2012-01-05 US disclosed
US-20120001154-A1 Aromatic amine derivative and organic electroluminescence device using the same IDEMITSU KOSAN CO., LTD. 2012-01-05 US disclosed
US-20070224448-A1 Organic Electroluminescent Device IDEMITSU KOSAN CO., LTD. (JP) 2007-09-27 US disclosed
US-20070224448-A1 Organic Electroluminescent Device IDEMITSU KOSAN CO., LTD. (JP) 2007-09-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190106391-A1 COMPOUNDS WITH SPIROBIFLUORENE-STRUCTURES TEC, NUDT1, DPYD AGTR1 788/4885CYP1A1 1403/4885CYP1A2 711/4885
US-20120001154-A1 Aromatic amine derivative and organic electroluminescence device using the same AOC3, NPR3, AOC2 AGTR1 951/4885CYP1A1 495/4885CYP1A2 684/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.