SCHEMBL27558474

SCHEMBL27558474

CC1(C(=O)O)C=C(c2c(F)cccc2I)C=C(C(=O)O)C1

nearest known ligand 0.33

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HCAR3 P49019 1/20 0.33
HCAR2 Q8TDS4 1/20 0.33
TTR P02766 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28185681 0.80 HCAR2 (0.34) HCAR3HCAR2TTR
SCHEMBL28046652 0.80 CA1 (0.36) HCAR3HCAR2TTR
SCHEMBL27775494 0.80 RARB (0.31)
SCHEMBL28056804 0.75 CA1 (0.39) HCAR2
SCHEMBL27775508 0.75 HCAR3 (0.36) HCAR3HCAR2
SCHEMBL27371651 0.74 BCL2L1 (0.38) HCAR3HCAR2
SCHEMBL19344710 0.71
SCHEMBL27459534 0.71
SCHEMBL28857964 0.70 ALDH1A1 (0.40) HCAR2
SCHEMBL28853255 0.70 TSHR (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102781942-A Disubstituted octahy-dropyrrolo [3,4-c]pyrroles as orexin receptor modulators JANSSEN PHARMACEUTICA NV 2012-11-14 CN disclosed
CN-1328247-C N-biphenylmethyl aminocycloalkanecarboxamide derivatives with a substiituent on the methyl useful as bradykinin antagonists MERCK & CO INC (US) 2007-07-25 CN disclosed
CN-1630633-A N-biphenylmethylaminocycloalkane carboxamide derivatives with substituents on the methyl group thereof as bradykinin antagonists MERCK & CO INC (US) 2005-06-22 CN disclosed