SCHEMBL27558917

SCHEMBL27558917

O=C(CCc1c(F)cccc1F)CCc1c(F)cccc1F

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 3/20 0.44
CES1 P23141 3/20 0.44
FFAR1 O14842 1/20 0.43
FFAR4 Q5NUL3 1/20 0.43
TAAR1 Q96RJ0 1/20 0.41
DAO P14920 1/20 0.41
MPO P05164 3/20 0.40
BCHE P06276 1/20 0.40
KDM4E B2RXH2 1/20 0.40
GAA P10253 1/20 0.38
IAPP P10997 1/20 0.38
NPC1 O15118 3/20 0.38
KMT2A Q03164 2/20 0.38
ALB P02768 1/20 0.38
MMP1 P03956 1/20 0.38
MMP2 P08253 1/20 0.38
MMP9 P14780 1/20 0.38
MMP12 P39900 1/20 0.38
POLB P06746 1/20 0.38
MAPT P10636 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19438660 0.84 MPO (0.54) CES2CES1FFAR1FFAR4TAAR1
SCHEMBL4714927 0.84 FFAR1 (0.59) CES2CES1FFAR1FFAR4KDM4E
SCHEMBL3937102 0.83 FFAR1 (0.40) CES2CES1FFAR1FFAR4TAAR1
SCHEMBL4717563 0.83 TAAR1 (0.42) CES2CES1FFAR1FFAR4TAAR1
SCHEMBL6158818 0.83 ALDH1A1 (0.50) CES2CES1FFAR1FFAR4TAAR1
SCHEMBL28805647 0.80 CES2 (0.40) CES2CES1FFAR1FFAR4BCHE
SCHEMBL6303011 0.78 MPO (0.39) CES2CES1FFAR1FFAR4TAAR1
SCHEMBL8979538 0.78 TP53 (0.51) GAANPC1KMT2APOLBRAB9A
SCHEMBL7701701 0.77 TAAR1 (0.52) CES2CES1TAAR1DAOKDM4E
SCHEMBL28159137 0.77 IAPP (0.46) CES2CES1FFAR4TAAR1MPO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105164113-B Pyrroloamide inhibitors 艾伯维公司 2018-03-02 CN disclosed
CN-104411709-B Can be used as imidazo [2, the 1] thiazole-3-ketone derivatives of the diagnostic agent of Alzheimer 霍夫曼-拉罗奇有限公司 2016-08-24 CN disclosed
CN-105164113-A Pyrroloamide inhibitors ABBVIE INC 2015-12-16 CN disclosed
CN-1349514-A Triazine derivatives having insecticidal activity SINGENTA PARTICIPATION AG (CH) 2002-05-15 CN disclosed