SCHEMBL27608010

SCHEMBL27608010

NOC(=O)[C@H](CCc1ccc2[nH]ccc2c1)C(=O)OCc1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 1/20 0.53
HDAC1 Q13547 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
CTNNB1 P35222 1/20 0.39
WNT3A P56704 1/20 0.39
SLC6A2 P23975 6/20 0.38
SLC6A4 P31645 6/20 0.38
SLC6A3 Q01959 6/20 0.38
FAAH O00519 1/20 0.38
MAPK14 Q16539 2/20 0.38
ROCK2 O75116 1/20 0.38
CYP19A1 P11511 1/20 0.37
NPC1 O15118 2/20 0.36
MAPT P10636 1/20 0.36
RAB9A P51151 1/20 0.36
AIMP2 Q13155 1/20 0.36
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA9 Q16790 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27607883 0.79 LNPEP (0.40) HDAC1SLC6A2SLC6A3RAB9ACA12
SCHEMBL27608029 0.78 ENPP2 (0.45) ENPP2SLC6A2SLC6A3MAPTMAOA
SCHEMBL27783442 0.76 FFAR4 (0.44)
SCHEMBL27643536 0.75 HTR1A (0.40) NPC1MAPTRAB9A
SCHEMBL27643798 0.74 KLK8 (0.35) SLC6A2SLC6A3CA12CA1CA2
SCHEMBL27689662 0.73 KMT2A (0.41) SLC6A2SLC6A3MAPTMAOB
SCHEMBL27767610 0.73 ALDH1A1 (0.46) SLC6A2SLC6A3CA12CA1CA2
SCHEMBL5326892 0.72 GRIK1 (0.60) ENPP2HDAC1HDAC8CTNNB1WNT3A
SCHEMBL188098 0.71 ENPP2 (0.60) ENPP2CTNNB1WNT3ASLC6A2SLC6A4
SCHEMBL6099420 0.71 NPC1 (0.55) ENPP2HDAC1HDAC8CTNNB1WNT3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100558428-C Calcitonin gene related peptide receptor antagonists BRISTOL MYERS SQUIBB CO (US) 2009-11-11 CN disclosed
CN-100558728-C Calcitonin gene related peptide receptor antagonists BRISTOL MYERS SQUIBB CO (US) 2009-11-11 CN disclosed
CN-1917921-A Calcitonin gene related peptide receptor antagonists BRISTOL MYERS SQUIBB CO (US) 2007-02-21 CN disclosed
CN-1671711-A Calcitonin gene related peptide receptor antagonists BRISTOL MYERS SQUIBB CO (US) 2005-09-21 CN disclosed