SCHEMBL27608908

SCHEMBL27608908

NCc1ccc(C(Cc2ccc(Cl)cc2)C(=O)c2cccnc2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.49
MAPT P10636 2/20 0.47
CYP2C9 P11712 2/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C19 P33261 1/20 0.46
GAA P10253 1/20 0.43
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
USP2 O75604 1/20 0.43
ALDH1A1 P00352 1/20 0.43
LMNA P02545 1/20 0.43
GPR132 Q9UNW8 1/20 0.42
KDM4E B2RXH2 1/20 0.42
HDAC1 Q13547 1/20 0.42
NPC1 O15118 1/20 0.41
PTPN1 P18031 1/20 0.41
POLB P06746 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6203529 0.89 TSHR (0.52) TSHRMAPTCYP2C9CYP1A2CYP3A4
SCHEMBL6204076 0.88 TSHR (0.49) TSHRMAPTCYP2C9CYP1A2CYP3A4
SCHEMBL6201072 0.81 TSHR (0.48) TSHRMAPTCYP2C9CYP1A2CYP3A4
SCHEMBL6201491 0.80 TSHR (0.50) TSHRMAPTCYP2C9CYP1A2CYP3A4
SCHEMBL6202599 0.77 PTPN1 (0.51) CYP2C9CYP2C19KMT2APTPN1
SCHEMBL6202785 0.73 NPC1 (0.46) TSHRMAPTCYP2C9CYP3A4CYP2C19
SCHEMBL10644705 0.72 NPC1 (0.52) TSHRMAPTCYP3A4CYP2C19GAA
SCHEMBL27628032 0.71 CHRM1 (0.60) TSHRGAAKMT2ALMNAPTPN1
SCHEMBL6204706 0.71 NPC1 (0.46) TSHRMAPTGAAMEN1KMT2A
SCHEMBL5263940 0.71 CNR1 (0.60) TSHRMAPTCYP2C9CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1681763-A Chemical compounds ASTRAZENECA AB (SE) 2005-10-12 CN disclosed