SCHEMBL6202599

SCHEMBL6202599

O=C(c1cccnc1)C(Cc1ccc(F)cc1)c1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 13/20 0.51
EPHX2 P34913 2/20 0.50
KMT2A Q03164 1/20 0.46
ATM Q13315 1/20 0.46
PTPN2 P17706 1/20 0.46
CHRM1 P11229 1/20 0.46
ECE1 P42892 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6203529 0.87 TSHR (0.52) PTPN1EPHX2KMT2ACHRM1ECE1
SCHEMBL27628032 0.82 CHRM1 (0.60) PTPN1EPHX2KMT2ACHRM1
SCHEMBL6203245 0.79 PSMB5 (0.44) PTPN1EPHX2
SCHEMBL27608839 0.78 PTPN1 (0.57) PTPN1PTPN2CHRM1
SCHEMBL27608908 0.77 TSHR (0.49) PTPN1KMT2ACYP2C9CYP2C19
SCHEMBL6204076 0.77 TSHR (0.49) KMT2ACYP2C9CYP2C19
SCHEMBL4664796 0.76 PPARA (0.56) PTPN1EPHX2CYP2C9CYP2C19
SCHEMBL6203944 0.75 EPHX1 (0.65) PTPN1ATMPTPN2CHRM1
SCHEMBL4197953 0.74 KCNA5 (0.50) CYP2C9CYP2C19
SCHEMBL6201072 0.74 TSHR (0.48) PTPN1KMT2ACYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050272036-A1 Ketones ASTRAZENECA AB (SE) 2005-12-08 US disclosed
CN-1681763-A Chemical compounds ASTRAZENECA AB (SE) 2005-10-12 CN disclosed
EP-1549600-A1 KETONES AstraZeneca AB (SE) 2005-07-06 EP disclosed
WO-2004011410-A1 CHEMICAL COMPOUNDS ASTRAZENECA AB (SE) 2004-02-05 WO disclosed