SCHEMBL6201072

SCHEMBL6201072

O=C(c1ccc(Cl)cc1)C(Cc1ccc(Cl)cc1)c1cccnc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.48
CYP19A1 P11511 1/20 0.48
KMT2A Q03164 3/20 0.47
ALOX15 P16050 1/20 0.47
MAPT P10636 1/20 0.46
NAMPT P43490 2/20 0.45
CNR1 P21554 1/20 0.45
CYP11B1 P15538 1/20 0.45
CYP11B2 P19099 1/20 0.45
PTPN1 P18031 2/20 0.44
MEN1 O00255 1/20 0.44
USP2 O75604 1/20 0.44
ALDH1A1 P00352 1/20 0.44
LMNA P02545 1/20 0.44
ADRB1 P08588 1/20 0.44
ADRB3 P13945 1/20 0.44
HAT1 O14929 1/20 0.43
EP300 Q09472 1/20 0.43
SLC1A3 P43003 1/20 0.43
SLC1A2 P43004 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6203529 0.87 TSHR (0.52) TSHRKMT2AMAPTCNR1PTPN1
SCHEMBL6204076 0.81 TSHR (0.49) TSHRCYP19A1KMT2AMAPTCNR1
SCHEMBL27608908 0.81 TSHR (0.49) TSHRKMT2AMAPTCNR1PTPN1
SCHEMBL6203634 0.80 NTSR1 (0.57) MAPTPTPN1LMNA
SCHEMBL8757592 0.79 CYP19A1 (0.54) TSHRCYP19A1KMT2AALOX15MAPT
SCHEMBL7144713 0.77 CYP19A1 (0.53) TSHRCYP19A1KMT2AALOX15MAPT
SCHEMBL6201491 0.77 TSHR (0.50) TSHRKMT2AALOX15MAPTNAMPT
SCHEMBL27628032 0.76 CHRM1 (0.60) TSHRKMT2APTPN1LMNA
Bromide SCHEMBL6284312 0.76 CYP19A1 (0.51) TSHRCYP19A1KMT2AALOX15MAPT
SCHEMBL8604244 0.75 CYP19A1 (0.57) TSHRCYP19A1MAPTCNR1ADRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050272036-A1 Ketones ASTRAZENECA AB (SE) 2005-12-08 US claimed
CN-1681763-A Chemical compounds ASTRAZENECA AB (SE) 2005-10-12 CN claimed
EP-1549600-A1 KETONES AstraZeneca AB (SE) 2005-07-06 EP claimed
WO-2004011410-A1 CHEMICAL COMPOUNDS ASTRAZENECA AB (SE) 2004-02-05 WO claimed
US-20050272036-A1 Ketones ASTRAZENECA AB (SE) 2005-12-08 US disclosed
CN-1681763-A Chemical compounds ASTRAZENECA AB (SE) 2005-10-12 CN disclosed
EP-1549600-A1 KETONES AstraZeneca AB (SE) 2005-07-06 EP disclosed
WO-2004011410-A1 CHEMICAL COMPOUNDS ASTRAZENECA AB (SE) 2004-02-05 WO disclosed