SCHEMBL6203529

SCHEMBL6203529

O=C(c1cccnc1)C(Cc1ccc(Cl)cc1)c1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.52
MAPT P10636 1/20 0.50
CNR1 P21554 1/20 0.48
PTPN1 P18031 9/20 0.48
CYP2C9 P11712 2/20 0.46
CYP2C19 P33261 2/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
GAA P10253 1/20 0.46
CHRM1 P11229 1/20 0.46
ECE1 P42892 1/20 0.45
EPHX2 P34913 1/20 0.45
MEN1 O00255 1/20 0.45
USP2 O75604 1/20 0.45
ALDH1A1 P00352 1/20 0.45
LMNA P02545 1/20 0.45
KMT2A Q03164 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6204076 0.89 TSHR (0.49) TSHRMAPTCNR1CYP2C9CYP2C19
SCHEMBL27608908 0.89 TSHR (0.49) TSHRMAPTCNR1PTPN1CYP2C9
SCHEMBL6202599 0.87 PTPN1 (0.51) PTPN1CYP2C9CYP2C19CHRM1ECE1
SCHEMBL6201072 0.87 TSHR (0.48) TSHRMAPTCNR1PTPN1CYP2C9
SCHEMBL6201491 0.82 TSHR (0.50) TSHRMAPTCYP2C9CYP2C19CYP1A2
SCHEMBL27628032 0.82 CHRM1 (0.60) TSHRPTPN1GAACHRM1EPHX2
SCHEMBL6202785 0.81 NPC1 (0.46) TSHRMAPTCYP2C9CYP2C19CYP3A4
SCHEMBL6203634 0.81 NTSR1 (0.57) MAPTPTPN1GAALMNA
SCHEMBL27608839 0.78 PTPN1 (0.57) PTPN1CYP3A4GAACHRM1ALDH1A1
SCHEMBL3370947 0.76 EPHX1 (0.56) CNR1CYP2C9CYP2C19EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050272036-A1 Ketones ASTRAZENECA AB (SE) 2005-12-08 US disclosed
CN-1681763-A Chemical compounds ASTRAZENECA AB (SE) 2005-10-12 CN disclosed
EP-1549600-A1 KETONES AstraZeneca AB (SE) 2005-07-06 EP disclosed
WO-2004011410-A1 CHEMICAL COMPOUNDS ASTRAZENECA AB (SE) 2004-02-05 WO disclosed