SCHEMBL6204076

SCHEMBL6204076

Cc1ccc(C(Cc2ccc(Cl)cc2)C(=O)c2cccnc2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.49
MAPT P10636 2/20 0.47
POLB P06746 2/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
KMT2A Q03164 5/20 0.43
MEN1 O00255 4/20 0.43
GAA P10253 1/20 0.43
FFAR2 O15552 1/20 0.43
USP2 O75604 1/20 0.43
ALDH1A1 P00352 1/20 0.43
LMNA P02545 1/20 0.43
CYP19A1 P11511 1/20 0.42
HCRTR2 O43614 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
CNR1 P21554 1/20 0.42
KDM4E B2RXH2 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6203529 0.89 TSHR (0.52) TSHRMAPTCYP1A2CYP3A4CYP2D6
SCHEMBL27608908 0.88 TSHR (0.49) TSHRMAPTPOLBCYP1A2CYP3A4
SCHEMBL6201072 0.81 TSHR (0.48) TSHRMAPTCYP1A2CYP3A4CYP2D6
SCHEMBL6201491 0.80 TSHR (0.50) TSHRMAPTPOLBCYP1A2CYP3A4
SCHEMBL6202599 0.77 PTPN1 (0.51) CYP2C9CYP2C19KMT2A
SCHEMBL10644705 0.75 NPC1 (0.52) TSHRMAPTCYP3A4CYP2C19KMT2A
SCHEMBL5263940 0.73 CNR1 (0.60) TSHRMAPTCYP1A2CYP3A4CYP2D6
SCHEMBL6202785 0.73 NPC1 (0.46) TSHRMAPTCYP3A4CYP2C9CYP2C19
SCHEMBL27628032 0.71 CHRM1 (0.60) TSHRKMT2AGAALMNA
SCHEMBL6204706 0.71 NPC1 (0.46) TSHRMAPTPOLBKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050272036-A1 Ketones ASTRAZENECA AB (SE) 2005-12-08 US disclosed
EP-1549600-A1 KETONES AstraZeneca AB (SE) 2005-07-06 EP disclosed
WO-2004011410-A1 CHEMICAL COMPOUNDS ASTRAZENECA AB (SE) 2004-02-05 WO disclosed