SCHEMBL2761271

SCHEMBL2761271

O=C(O)Nc1c(-c2ccccc2)noc1-c1ccc(Br)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LPAR1 Q92633 3/20 0.48
LPAR3 Q9UBY5 1/20 0.48
PTGS1 P23219 1/20 0.48
KMT2A Q03164 3/20 0.45
KDM4E B2RXH2 2/20 0.44
HTT P42858 2/20 0.44
MEN1 O00255 2/20 0.44
ALDH1A1 P00352 1/20 0.44
HKDC1 Q2TB90 1/20 0.44
MCOLN3 Q8TDD5 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
MAPT P10636 1/20 0.43
TSHR P16473 1/20 0.43
RAB9A P51151 1/20 0.42
ABCC3 O15438 1/20 0.41
ABCC4 O15439 1/20 0.41
ABCB11 O95342 1/20 0.41
CYP2C8 P10632 1/20 0.41
CYP2C9 P11712 1/20 0.41
ABCB4 P21439 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12973608 0.82 LPAR1 (0.72) LPAR1LPAR3PTGS1ALDH1A1RAB9A
SCHEMBL6003 0.81 LPAR1 (0.54) LPAR1LPAR3KMT2AKDM4EHTT
SCHEMBL9903838 0.81 NPSR1 (0.48) KMT2AKDM4EHTTMEN1ALDH1A1
SCHEMBL2761396 0.78 PTGS1 (0.58) PTGS1KMT2AKDM4EHTTMEN1
SCHEMBL4304 0.78 RAB9A (0.40) LPAR1LPAR3KMT2AKDM4EHTT
SCHEMBL4029460 0.76 NPSR1 (0.61) PTGS1KMT2AKDM4EHTTMEN1
SCHEMBL4035675 0.76 MAPT (0.67) LPAR1LPAR3PTGS1KMT2AKDM4E
SCHEMBL19742000 0.74 PTGS2 (0.51) PTGS1KMT2AMEN1ALDH1A1NR1H4
SCHEMBL2761365 0.73 PTGS1 (0.62) PTGS1KMT2AKDM4EHTTMEN1
SCHEMBL4034308 0.72 KDM4E (0.49) LPAR1LPAR3PTGS1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010141768-A2 POLYCYCLIC ANTAGONISTS OF LYSOPHOSPHATIDIC ACID RECEPTORS AMIRA PHARMACEUTICALS, INC. (US) 2010-12-09 WO disclosed