SCHEMBL27633952

SCHEMBL27633952

CCOS(=O)(=O)c1ccc(C)c(C2CC2)c1

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HTT P42858 3/20 0.39
HRH4 Q9H3N8 5/20 0.36
HTR6 P50406 6/20 0.36
ALDH1A1 P00352 2/20 0.35
HCRTR2 O43614 1/20 0.33
TSHR P16473 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29024319 0.88 CA2 (0.36) HTTHRH4HTR6ALDH1A1TSHR
SCHEMBL28759659 0.83 HTT (0.33) HTT
SCHEMBL28252743 0.80 HTT (0.33) HTTALDH1A1HCRTR2
SCHEMBL7067658 0.78 ALDH1A1 (0.41) HTTHTR6ALDH1A1TSHRSMN1; SMN2
SCHEMBL28966886 0.77 HTT (0.37) HTTALDH1A1TDP1
SCHEMBL28645585 0.77 PTPN1 (0.40) HTTALDH1A1TSHRSMN1; SMN2TDP1
SCHEMBL29104732 0.77 CA1 (0.41) HTTALDH1A1TSHRTDP1
SCHEMBL28211544 0.76 KMT2A (0.38) HTTALDH1A1TSHR
SCHEMBL8788235 0.75 CYP2D6 (0.37) HTTALDH1A1HCRTR2TSHR
SCHEMBL6754204 0.74 LMNA (0.41) HTTALDH1A1TSHRSMN1; SMN2TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108602813-A Heteroaryl hydroxypyrimidinone as apj receptor agonist 百时美施贵宝公司 2018-09-28 CN disclosed
CN-103664973-A Spiro-oxindole compounds and their use as therapeutic agents XENON PHARMACEUTICALS INC 2014-03-26 CN disclosed
CN-102600162-A Pyridazine derivatives and their use as therapeutic agents XENON PHARMACEUTICALS INC 2012-07-25 CN disclosed
CN-102256983-A Spirooxindole compounds and their use as therapeutic agents XENON PHARMACEUTICALS INC 2011-11-23 CN disclosed
CN-101980709-A Pyridazine derivatives and their use as therapeutic agents XENON PHARMACEUTICALS INC 2011-02-23 CN disclosed
CN-101669952-A Pyridazine derivatives and their use as therapeutic agents XENON PHARMACEUTICALS INC 2010-03-17 CN disclosed
CN-100558713-C Pyridazine derivatives and their use as therapeutic agents XENON PHARMACEUTICALS INC (CA) 2009-11-11 CN disclosed
CN-101160289-A Pyridazine derivatives and their use as therapeutic agents XENON PHARMACEUTICALS INC (CA) 2008-04-09 CN disclosed
CN-101090724-A Pyridine derivatives for inhibiting human stearoyl-CoA desaturase XENON PHARMACEUTICALS INC (CA) 2007-12-19 CN disclosed
CN-1829698-A Pyridazine derivatives and their use as therapeutic agents XENON PHARMACEUTICALS INC (CA) 2006-09-06 CN disclosed