SCHEMBL27658652

SCHEMBL27658652

CN(C[SH](=O)=O)c1ncc(-c2cc(Cl)ccc2O)cn1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 5/20 0.37
VEGFA P15692 1/20 0.37
FLT1 P17948 1/20 0.37
EGLN1 Q9GZT9 1/20 0.37
KDM4E B2RXH2 3/20 0.35
LMNA P02545 3/20 0.35
NPC1 O15118 2/20 0.35
CASP3 P42574 2/20 0.35
CDK9 P50750 2/20 0.35
RAB9A P51151 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
SENP7 Q9BQF6 2/20 0.35
NFKB1 P19838 1/20 0.35
CDK5 Q00535 1/20 0.35
NFKB2 Q00653 1/20 0.35
RELA Q04206 1/20 0.35
CDK5R1 Q15078 1/20 0.35
SENP8 Q96LD8 1/20 0.35
SENP6 Q9GZR1 1/20 0.35
PIM1 P11309 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2110554 0.76 IDO1 (0.39) IDO1VEGFAFLT1EGLN1KDM4E
SCHEMBL2111844 0.70 PDK1 (0.45) VEGFAFLT1EGLN1KDM4ELMNA
SCHEMBL2113204 0.69 ALDH1A1 (0.43) LMNACDK9SMN1; SMN2MEN1KMT2A
SCHEMBL14832716 0.69 FTO (0.45) IDO1KDM4EPIM1EPHX2MEN1
SCHEMBL2113926 0.69 TRPM8 (0.39) LMNACDK9HTTCYP1A2CYP3A4
SCHEMBL2112842 0.66 IDO1 (0.54) IDO1LMNASMN1; SMN2PIM1EPHX2
SCHEMBL1753343 0.66 PTGDR2 (0.64) MAPTTDP1
SCHEMBL28180078 0.65 SLC6A7 (0.31) CYP2D6CYP2C19SLC6A7
SCHEMBL1743707 0.64 DYRK1A (0.44) IDO1LMNAPIM1EPHX2MAPT
SCHEMBL1093987 0.64 DYRK1A (0.44) IDO1LMNAPIM1EPHX2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100575330-C Novel compounds ASTRAZENECA AB 2009-12-30 CN claimed
CN-1791572-A Novel compounds ASTRAZENECA AB (SE) 2006-06-21 CN claimed
CN-100575330-C Novel compounds ASTRAZENECA AB 2009-12-30 CN disclosed
CN-1791572-A Novel compounds ASTRAZENECA AB (SE) 2006-06-21 CN disclosed