SCHEMBL27675110

SCHEMBL27675110

O=C(O)c1cn(C(=O)Nc2cccc(SC(F)(F)F)c2)c2ccccc2c1=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 3/20 0.46
DRD2 P14416 2/20 0.43
TRPV1 Q8NER1 5/20 0.42
CREBBP Q92793 2/20 0.42
EP300 Q09472 1/20 0.42
RXFP1 Q9HBX9 3/20 0.42
UBE2M P61081 1/20 0.41
DCUN1D1 Q96GG9 1/20 0.41
MAOB P27338 1/20 0.40
S1PR1 P21453 1/20 0.39
S1PR3 Q99500 1/20 0.39
LMNA P02545 2/20 0.39
KCNK2 O95069 1/20 0.39
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.39
USP2 O75604 1/20 0.39
ALDH1A1 P00352 1/20 0.39
HPGD P15428 1/20 0.39
TSHR P16473 1/20 0.39
HTT P42858 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27675189 0.84 GRIK1 (0.51) CREBBPRXFP1LMNAMEN1HTT
SCHEMBL27693487 0.82 LMNA (0.51) CHRM1CREBBPEP300MAOBLMNA
SCHEMBL27675195 0.82 CFD (0.49)
SCHEMBL27693567 0.82 CREBBP (0.47) CHRM1CREBBPEP300MAOBLMNA
SCHEMBL27693586 0.81 MAOB (0.60) CHRM1CREBBPEP300RXFP1MAOB
SCHEMBL27675227 0.81 CFTR (0.48) CHRM1CREBBPEP300MAOBLMNA
SCHEMBL27675196 0.81 CREBBP (0.52) CHRM1CREBBPEP300MAOBLMNA
SCHEMBL27675320 0.80 ALDH1A1 (0.46) CHRM1CREBBPEP300S1PR1S1PR3
SCHEMBL27693516 0.80 CREBBP (0.61) CREBBPEP300RXFP1MAOBKDM4E
SCHEMBL27675135 0.80 CREBBP (0.54) CHRM1CREBBPEP300MAOBLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101006076-B Modulators of ATP-binding cassette transporters VERTEX PHARMA 2010-09-29 CN disclosed
CN-101006076-A Modulators of ATP-binding cassette transporters VERTEX PHARMA (US) 2007-07-25 CN disclosed